Substituted N-heterocyclyl-and N-heteroaryltetrahydropyrimidines and their salts and their use as herbicidal active substances
阅读说明：本技术 取代的n-杂环基-和n-杂芳基四氢嘧啶酮及其盐，以及其作为除草活性物质的用途 (Substituted N-heterocyclyl-and N-heteroaryltetrahydropyrimidines and their salts and their use as herbicidal active substances ) 是由 J·施密特 H·赫尔姆克 J·弗拉肯波尔 A·M·莱因格鲁伯 T·穆勒 E·阿斯马斯 E 于 2018-12-17 设计创作，主要内容包括：本发明涉及通式(I)的取代的N-杂环基-和N-杂芳基四氢嘧啶酮或其盐,其中通式(I)中的基团如说明书中所定义,以及涉及其作为除草剂、特别是用于防治栽培植物作物中的杂草和/或禾本科杂草,和/或作为植物生长调节剂用于影响栽培植物作物的生长的用途。<Image he="289" wi="414" file="DDA0002636287970000011.GIF" imgContent="drawing" imgFormat="GIF" orientation="portrait" inline="no"></Image>(The invention relates to substituted N-heterocyclyl-and N-heteroaryltetrahydropyrimidinone compounds of general formula (I) or salts thereof, wherein the radicals in the general formula (I) are as defined in the description, and to the use thereof as herbicides, in particular for controlling weeds and/or grasses in crops of cultivated plants, and/or as plant growth regulators for influencing the growth of crops of cultivated plants.)
1. Substituted N-heterocyclyl-or N-heteroaryltetrahydropyrimidinone of the general formula (I) and/or its salts
Wherein
Q represents a group Q-1 to Q-30
Wherein the arrows represent the bond of the respective Q group to the nitrogen of the tetrahydropyrimidinone of the general formula (I),
A1、A2、A3、A4identical or different and, independently of one another, represent N (nitrogen) or a moiety C-R8But the number of adjacent nitrogen atoms is by no means more than two, and according to the definition below,wherein moiety C-R8R of (A) to (B)8In each case having the same or different meanings, or
A1And A2When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A2And A3When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A3And A4When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted,
R1represents hydrogen, hydroxy, (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkyl, (C)1-C8) -hydroxyalkyl, hydroxycarbonyl- (C)1-C8) Alkylene group, (C)1-C8) -alkoxy, (C)1-C8) -alkoxy- (C)1-C8) Alkylene group, (C)1-C8) Alkoxy-alkoxy (C)1-C8) -haloalkoxy, (C)3-C10) -cycloalkyl, (C)3-C10) Halocycloalkyl, aryl, heteroaryl, (C)3-C10) -cycloalkyl- (C)1-C8) Alkylene, heterocyclic, (C)2-C8) -alkenyl, (C)2-C8) -alkenyloxy, (C)2-C8) -alkynyl, (C)2-C8) -alkynyloxy, amino, bis [ (C)1-C8) -alkyl radical]Amino, aryl- (C)1-C8) Alkylene, heteroaryl- (C)1-C8) Alkylene, heterocyclyl- (C)1-C8) Alkylene group, (C)1-C8) Cyanoalkyl, C (O) R12、C(O)OR12、C(O)NR10R11、SO2R13、R12O(O)C-(C1-C8) Alkylene, arylcarbonyl- (C)1-C8) Alkylene group, (C)1-C8) -alkylcarbonyl- (C)1-C8) Alkylene, heteroarylcarbonyl- (C)1-C8) Alkylene, heterocyclylcarbonyl- (C)1-C8) Alkylene group, (C)1-C7) -alkylcarbonyloxy- (C)1-C8) -an alkylene group,
R2and R9Independently of one another, represents hydrogen, hydroxy, halogen, (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkyl, (C)3-C10) Cycloalkyl, aryl, heteroaryl, heterocyclyl, aryl- (C) 1-C8) -alkyl, heteroaryl- (C)1-C8) Alkyl, heterocyclyl- (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyl, (C)2-C8) -alkynyl, arylcarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylcarbonyl- (C)1-C8) -alkyl, heteroarylcarbonyl- (C)1-C8) Alkyl radicals, (C)3-C10) -cycloalkylcarbonyl- (C)1-C8) Alkyl, aryl- (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxy- (C)1-C8) Alkyl, arylcarbonyloxy- (C)1-C8) Alkyl, heteroarylcarbonyloxy- (C)1-C8) Alkyl, heterocyclylcarbonyloxy- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylcarbonyloxy- (C)1-C8) Alkyl radicals, (C)3-C8) -cycloalkylcarbonyloxy- (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkoxy- (C)1-C8) Alkyl, arylRadical- (C)1-C8) -alkoxy- (C)1-C8) -alkyl, heteroaryl- (C)1-C8) -alkoxy- (C)1-C8) Alkyl, C (O) R12、C(O)OR12、C(O)NR10R11、OR12、SR13、SOR13、SO2R13、NR10R11、R10R11N-(C1-C8) -alkyl, cyano- (C)1-C8) -alkyl, hydroxycarbonyl- (C)1-C8) Alkyl, hydroxycarbonyl, aminocarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylaminocarbonyl- (C)1-C8) Alkyl radicals, (C)3-C8) -cycloalkylaminocarbonyl- (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyloxycarbonyl- (C)1-C8) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl, cyano, hydroxy- (C)1-C8) -alkyl, or
R1And R2Together with the nitrogen or carbon atom to which they are respectively attached form a fully or partially saturated ring having a total of 3 to 7 members, said ring being optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted, or
R2And R9Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R3represents hydroxy, mercapto, halogen, NR10R11、(C1-C8) -alkoxy, (C)3-C10) -cycloalkyl- (C)1-C8) Alkoxy, aryl- (C)1-C8) -alkoxy, (C)1-C8) -alkoxy- (C)1-C8) -alkoxy, arylcarbonyloxy, (C)1-C8) -alkylcarbonyloxy, (C)1-C8) -alkoxy- (C)1-C8) -alkylcarbonyloxy, aryl- (C)1-C8) -alkylcarbonyloxy, heteroarylcarbonyloxy, (C)3-C10) -cycloalkylcarbonyloxy, heterocyclylcarbonyloxy, (C)1-C8) -haloalkylcarbonyloxy, (C)2-C8) Alkenylcarbonyloxy, OC (O) OR12、OC(O)SR13、OC(S)OR12、OC(S)SR13、OSO2R13、OSO2OR12、OCHO，
R4And R7Independently of one another, represents hydrogen, mercapto, hydroxy, halogen, (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkyl, (C)3-C10) -cycloalkyl, (C)3-C10) -cycloalkyl- (C)1-C8) Alkyl, aryl, heteroaryl, heterocyclyl, aryl- (C)1-C8) -alkyl, heteroaryl- (C)1-C8) Alkyl, heterocyclyl- (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyl, (C)2-C8) -alkynyl, (C)2-C8) -haloalkenyl, (C)2-C8) -haloalkynyl, (C)3-C10) -halocycloalkyl, (C)4-C10) Cycloalkenyl radical, (C)4-C10) Halocycloalkenyl, aryl- (C)2-C8) -alkenyl, heteroaryl- (C) 2-C8) -alkenyl, heterocyclyl- (C)2-C8) -alkenyl, aryl- (C)2-C8) -alkynyl, heteroaryl- (C)2-C8) -alkynyl, heterocyclyl- (C)2-C8) -alkynyl, (C)3-C10) -cycloalkyl- (C)2-C8) -alkynyl, arylcarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylcarbonyl- (C)1-C8) -alkyl, heteroarylcarbonyl- (C)1-C8) Alkyl radicals, (C)3-C10) -cycloalkylcarbonyl- (C)1-C8) Alkyl, aryl- (C)1-C8) -alkanesOxycarbonyl radical- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxy- (C)1-C8) Alkyl, arylcarbonyloxy- (C)1-C8) Alkyl, heteroarylcarbonyloxy- (C)1-C8) Alkyl, heterocyclylcarbonyloxy- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylcarbonyloxy- (C)1-C8) Alkyl radicals, (C)3-C8) -cycloalkylcarbonyloxy- (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkoxy- (C)1-C8) Alkyl, aryl- (C)1-C8) -alkoxy- (C)1-C8) -alkyl, heteroaryl- (C)1-C8) -alkoxy- (C)1-C8) Alkyl, CHO, C (O) R12、C(O)OR12、C(O)NR10R11、OR12、SR13、SOR13、SO2R13、NR10R11、R10R11N-(C1-C8) -alkyl, cyano- (C)1-C8) -alkyl, hydroxycarbonyl- (C)1-C8) -alkyl, hydroxycarbonyl, (C)1-C8) -haloalkoxy- (C)1-C8) Alkylthio group(s), (C)1-C8) -alkylthio- (C)1-C8) Alkylene group, (C)1-C8) -haloalkylthio- (C)1-C8) Alkylthio group(s), (C)1-C8) -alkylthio- (C)1-C8) Alkylthio, aminocarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylaminocarbonyl- (C)1-C8) Alkyl radicals, (C)3-C8) -cycloalkylaminocarbonyl- (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyloxycarbonyl- (C) 1-C8) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl, cyano, hydroxy- (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyloxy- (C)1-C8) -alkyl, or
When Q represents Q-3, Q-4, Q-8, Q-9, Q-12 and Q-19, R4And R7Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R5represents hydrogen, formyl or (C)1-C8) Alkyl radicals, (C)1-C8) Haloalkyl, hydroxy- (C)1-C8) -alkyl, hydroxycarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxy- (C)1-C8) Alkyl radicals, (C)3-C10) -cycloalkyl, (C)3-C10) Halocycloalkyl, aryl, heteroaryl, (C)3-C10) -cycloalkyl- (C)1-C8) Alkyl, heterocyclyl, (C)2-C8) -alkenyl, (C)2-C8) -alkynyl, NR10R11Aryl group- (C)1-C8) -alkyl, heteroaryl- (C)1-C8) Alkyl, heterocyclyl- (C)1-C8) Alkyl radicals, (C)1-C8) Cyanoalkyl, C (O) R12、C(O)OR12、C(O)NR10R11、SO2R13、(C1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyloxycarbonyl- (C)1-C8) Alkyl, aryl- (C)1-C8) -alkoxycarbonyl- (C)1-C8) -alkyl, heteroaryl- (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl, aryloxy carbonyl- (C)1-C8) -alkyl, arylcarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylcarbonyl- (C)1-C8) -alkyl, heteroarylcarbonyl- (C) 1-C8) -alkyl, heterocyclylcarbonyl- (C)1-C8) -alkyl, or
When Q represents Q-13, Q-14, Q-15, Q-25 and Q-26, R4And R5Together with the nitrogen or carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R6represents hydrogen or (C)1-C8) -an alkyl group,
R8represents hydrogen, halogen, cyano, nitro, mercapto, hydroxy, NR10R11、OR12、SR13、SOR13、SO2R13Thiocyanato, isothiocyanato, formyl, (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyl, (C)2-C8) -alkynyl, (C)1-C10) -haloalkyl, (C)2-C8) -haloalkenyl, (C)2-C8) -haloalkynyl, (C)3-C10) -cycloalkyl, (C)3-C10) -halocycloalkyl, (C)4-C10) Cycloalkenyl radical, (C)4-C10) Halocycloalkenyl, pentafluorothio, (C)1-C8) -alkoxy- (C)1-C8) -haloalkyl, (C)1-C8) -haloalkoxy- (C)1-C8) -haloalkyl, (C)1-C8) -haloalkoxy- (C)1-C8) Alkyl, aryl- (C)1-C8) Alkyl, heteroaryl- (C)1-C8) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C8) Alkyl radicals, (C)4-C10) -cycloalkenyl- (C)1-C8) Alkyl, heterocyclyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxy- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylthio- (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkylthio- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylcarbonyl- (C) 1-C8) Alkyl, C (O) OR12、C(O)NR10R11、C(O)R12、-C＝NOR12、-C＝NOH、R10R11N-(C1-C8) -alkyl, R12O(O)C-(C1-C8) Alkyl, hydroxycarbonyl- (C)1-C8) Alkyl, aryl- (C)1-C8) -alkynyl, heteroaryl- (C)1-C8) -alkynyl, heterocyclyl- (C)1-C8) -alkynyl, tris [ (C)1-C8) -alkyl radical]Silyl radical- (C)2-C8) -alkynyl, bis [ (C)1-C8) -alkyl radical](aryl) silyl- (C)2-C8) -alkynyl, diaryl [ (C)1-C8) -alkyl radical]Silyl radical- (C)2-C8) -alkynyl, (C)3-C8) -cycloalkyl- (C)2-C8) -alkynyl, aryl- (C)2-C8) -alkenyl, heteroaryl- (C)2-C8) -alkenyl, heterocyclyl- (C)2-C8) -alkenyl, (C)3-C8) -cycloalkyl- (C)2-C8) -alkenyl, (C)1-C8) -alkoxy- (C)1-C8) -alkoxy- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylaminosulfonamido, (C)3-C8) -cycloalkylaminosulfonylamino, diazo, aryldiazo, tris [ (C)1-C8) -alkyl radical]Silyl, bis [ (C)1-C8) -alkyl radical](aryl) silyl, diaryl [ (C)1-C8) -alkyl radical]A silyl group (a) having a silyl group (a),
R10and R11Are identical or different and independently of one another represent hydrogen, (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyl, (C)2-C8) -alkynyl, (C)1-C8) Cyanoalkyl, (C)1-C10) -haloalkyl, (C)2-C8) -haloalkenyl, (C)2-C8) -haloalkynyl, (C)3-C10) -cycloalkyl, (C)3-C10) -halocycloalkyl, (C)4-C10) Cycloalkenyl radical, (C)4-C10) -halocycloalkenyl radical, (C)1-C8) -alkoxy- (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkoxy- (C)1-C8) Alkyl radicals, (C)1-C8) -alkylthio- (C)1-C8) Alkyl radicals, (C)1-C8) -haloalkylthio- (C) 1-C8) Alkyl radicals, (C)1-C8) -alkoxy- (C)1-C8) Haloalkyl, aryl- (C)1-C8) Alkyl, heteroaryl- (C)1-C8) Alkyl radicals, (C)3-C10) -cycloalkyl- (C)1-C8) Alkyl radicals, (C)4-C10) -cycloalkenyl- (C)1-C8) Alkyl radical, COR12、SO2R13、(C1-C8) -alkyl-HNO2S-、(C3-C10) -cycloalkyl-HNO2S-, heterocyclic group, (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl radicals, (C)1-C8) Alkoxycarbonyl, aryl- (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl, aryl- (C)1-C8) Alkoxycarbonyl, heteroaryl- (C)1-C8) Alkoxycarbonyl, (C)2-C8) -alkenyloxycarbonyl, (C)2-C8) -alkynyloxycarbonyl, heterocyclyl- (C)1-C8) -an alkyl group,
R12is represented by (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyl, (C)2-C8) -alkynyl, (C)1-C8) Cyanoalkyl, (C)1-C10) -haloalkyl, (C)2-C8) -haloalkenyl, (C)2-C8) -haloalkynyl, (C)3-C10) -cycloalkyl, (C)3-C10) -halocycloalkyl, (C)4-C10) Cycloalkenyl radical, (C)4-C10) -halocycloalkenyl radical, (C)1-C8) -alkoxy- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxy- (C)1-C8) Haloalkyl, aryl- (C)1-C8) Alkyl, heteroaryl- (C)1-C8) Alkyl radicals, (C)3-C10) -cycloalkyl- (C)1-C8) Alkyl radicals, (C)4-C10) -cycloalkenyl- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxycarbonyl- (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyloxycarbonyl- (C)1-C8) Alkyl, aryl- (C)1-C8) -alkoxycarbonyl- (C)1-C8) -alkyl, hydroxycarbonyl- (C)1-C8) Alkyl, heterocyclyl- (C)1-C8) -an alkyl group,
R13Is represented by (C)1-C8) Alkyl radicals, (C)2-C8) -alkenyl, (C)2-C8) -alkynyl, (C)1-C8) Cyanoalkyl, (C)1-C10) -haloalkyl, (C)2-C8) -haloalkenyl, (C)2-C8) -haloalkynyl, (C)3-C10) -cycloalkyl, (C)3-C10) -halocycloalkyl, (C)4-C10) Cycloalkenyl radical, (C)4-C10) -halocycloalkenyl radical, (C)1-C8) -alkoxy- (C)1-C8) Alkyl radicals, (C)1-C8) -alkoxy- (C)1-C8) Haloalkyl, aryl- (C)1-C8) Alkyl, heteroaryl- (C)1-C8) Alkyl, heterocyclyl- (C)1-C8) Alkyl radicals, (C)3-C10) -cycloalkyl- (C)1-C8) Alkyl radicals, (C)4-C10) -cycloalkenyl- (C)1-C8) Alkyl, NR10R11，
R14And R15Independently of one another, represents hydrogen, (C)1-C8) -alkyl, halogen, or
R9And R15Together with the carbon atoms to which they are each attached form a ring having a total of 3 to 7A fully or partially saturated ring of members, said ring optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
and
w represents oxygen.
2. A compound of the general formula (I) and/or a salt thereof as claimed in claim 1, characterized in that
Q represents a group Q-1 to Q-30
Wherein the arrows represent the bond of the respective Q group to the nitrogen of the tetrahydropyrimidinone of the general formula (I),
A1、A2、A3、A4identical or different and, independently of one another, represent N (nitrogen) or a moiety C-R8But no more than two adjacent nitrogen atoms and according to the definition below, wherein the moiety C-R 8R of (A) to (B)8In each case having the same or different meanings, or
A1And A2When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A2And A3When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A3And A4When each is a group C-R8When they are combined with the atoms to which they are attached form a fully saturated moietyA partially saturated or fully unsaturated 5 to 7 membered ring, said ring optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted,
R1represents hydrogen, hydroxy, (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkyl, (C)1-C7) -hydroxyalkyl, hydroxycarbonyl- (C)1-C7) Alkylene group, (C)1-C7) -alkoxy, (C)1-C7) -alkoxy- (C)1-C7) Alkylene group, (C)1-C7) Alkoxy-alkoxy (C)1-C7) -haloalkoxy, (C)3-C8) -cycloalkyl, (C)3-C8) Halocycloalkyl, aryl, heteroaryl, (C) 3-C8) -cycloalkyl- (C)1-C7) Alkylene, heterocyclic, (C)2-C7) -alkenyl, (C)2-C7) -alkenyloxy, (C)2-C7) -alkynyl, (C)2-C7) -alkynyloxy, amino, bis [ (C)1-C7) -alkyl radical]Amino, aryl- (C)1-C7) Alkylene, heteroaryl- (C)1-C7) Alkylene, heterocyclyl- (C)1-C7) Alkylene group, (C)1-C7) Cyanoalkyl, C (O) R12、C(O)OR12、C(O)NR10R11、SO2R13、R12O(O)C-(C1-C7) Alkylene, arylcarbonyl- (C)1-C7) Alkylene group, (C)1-C7) -alkylcarbonyl- (C)1-C7) Alkylene, heteroarylcarbonyl- (C)1-C7) Alkylene, heterocyclylcarbonyl- (C)1-C7) Alkylene group, (C)1-C7) -alkylcarbonyloxy- (C)1-C7) -an alkylene group,
R2and R9Independently of one another, represents hydrogen, hydroxy, halogen, (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkyl, (C)3-C8) Cycloalkyl, aryl, heteroaryl, heterocyclyl, aryl- (C)1-C7) -alkyl, heteroaryl- (C)1-C7) Alkyl, heterocyclyl- (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyl, (C)2-C7) -alkynyl, (C)1-C7) -alkoxy- (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkoxy- (C)1-C7) Alkyl, aryl- (C)1-C7) -alkoxy- (C)1-C7) -alkyl, heteroaryl- (C)1-C7) -alkoxy- (C)1-C7) -alkyl, OR12、SR13、SOR13、SO2R13、NR10R11、R10R11N-(C1-C7) -alkyl, cyano- (C)1-C7) Alkyl, cyano, hydroxy- (C)1-C7) -alkyl, or
R1And R2Together with the nitrogen or carbon atom to which they are respectively attached form a fully or partially saturated ring having a total of 3 to 7 members, said ring being optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted, or
R2And R9Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R3represents hydroxy, mercapto, halogen, NR10R11、(C1-C7) -alkoxy, (C)3-C8) -cycloalkyl- (C)1-C7) Alkoxy, aryl- (C)1-C7) -alkoxy, (C)1-C7) -alkoxy- (C)1-C7) -alkoxy, arylcarbonyloxy, (C)1-C7) -alkylcarbonyloxy, (C)1-C7) -alkoxy- (C)1-C7) -alkylcarbonyloxy, aryl- (C)1-C7) -alkylcarbonyloxy, heteroarylcarbonyloxy, (C)3-C8) -cycloalkanesAlkylcarbonyloxy, heterocyclylcarbonyloxy, (C)1-C7) -haloalkylcarbonyloxy, (C)2-C7) Alkenylcarbonyloxy, OC (O) OR12、OC(O)SR13、OC(S)OR12、OC(S)SR13、OSO2R13、OSO2OR12、OCHO，
R4And R7Independently of one another, represents hydrogen, mercapto, hydroxy, halogen, (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkyl, (C)3-C8) -cycloalkyl, (C)3-C8) -cycloalkyl- (C)1-C7) Alkyl, aryl, heteroaryl, heterocyclyl, aryl- (C)1-C7) -alkyl, heteroaryl- (C)1-C7) Alkyl, heterocyclyl- (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyl, (C)2-C7) -alkynyl, (C)2-C7) -haloalkenyl, (C)2-C7) -haloalkynyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) Halocycloalkenyl, aryl- (C)2-C7) -alkenyl, heteroaryl- (C) 2-C7) -alkenyl, heterocyclyl- (C)2-C7) -alkenyl, aryl- (C)2-C7) -alkynyl, heteroaryl- (C)2-C7) -alkynyl, heterocyclyl- (C)2-C7) -alkynyl, (C)3-C8) -cycloalkyl- (C)2-C7) -alkynyl, arylcarbonyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylcarbonyl- (C)1-C7) -alkyl, heteroarylcarbonyl- (C)1-C7) Alkyl radicals, (C)3-C8) -cycloalkylcarbonyl- (C)1-C7) Alkyl, aryl- (C)1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkoxy- (C)1-C7) Alkyl, arylcarbonyloxy- (C)1-C7) Alkyl, heteroarylcarbonyloxy- (C)1-C7) Alkyl, heterocyclylcarbonyloxy- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylcarbonyloxy- (C)1-C7) Alkyl radicals, (C)3-C7) -cycloalkylcarbonyloxy- (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkoxy- (C)1-C7) Alkyl, aryl- (C)1-C7) -alkoxy- (C)1-C7) -alkyl, heteroaryl- (C)1-C7) -alkoxy- (C)1-C7) Alkyl, CHO, C (O) R12、C(O)OR12、C(O)NR10R11、OR12、SR13、SOR13、SO2R13、NR10R11、R10R11N-(C1-C7) -alkyl, cyano- (C)1-C7) -alkyl, hydroxycarbonyl- (C)1-C7) -alkyl, hydroxycarbonyl, (C)1-C7) -haloalkoxy- (C)1-C7) Alkylthio group(s), (C)1-C7) -alkylthio- (C)1-C7) Alkylene group, (C)1-C7) -haloalkylthio- (C)1-C7) Alkylthio group(s), (C)1-C7) -alkylthio- (C)1-C7) Alkylthio, aminocarbonyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylaminocarbonyl- (C)1-C7) Alkyl radicals, (C)3-C7) -cycloalkylaminocarbonyl- (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyloxycarbonyl- (C) 1-C7) Alkyl radicals, (C)3-C7) -cycloalkyl- (C)1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl, cyano, hydroxy- (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyloxy- (C)1-C7) -alkyl, or
When Q represents Q-3, Q-4, Q-8, Q-9, Q-12, Q-13, Q-19 and Q-30, R4And R7And each of themFrom the attached carbon atoms together form a fully or partially saturated ring having a total of 3 to 7 members, said ring optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R5represents hydrogen, formyl or (C)1-C7) Alkyl radicals, (C)1-C7) Haloalkyl, hydroxy- (C)1-C7) -alkyl, hydroxycarbonyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkoxy- (C)1-C7) Alkyl radicals, (C)3-C8) -cycloalkyl, (C)3-C8) Halocycloalkyl, aryl, heteroaryl, (C)3-C8) -cycloalkyl- (C)1-C7) Alkyl, heterocyclyl, (C)2-C7) -alkenyl, (C)2-C7) -alkynyl, NR10R11Aryl group- (C)1-C7) -alkyl, heteroaryl- (C)1-C7) Alkyl, heterocyclyl- (C)1-C7) Alkyl radicals, (C)1-C7) Cyanoalkyl, C (O) R12、C(O)OR12、C(O)NR10R11、SO2R13、(C1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyloxycarbonyl- (C)1-C7) Alkyl, aryl- (C)1-C7) -alkoxycarbonyl- (C)1-C7) -alkyl, heteroaryl- (C)1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl, aryloxy carbonyl- (C)1-C7) -alkyl, arylcarbonyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylcarbonyl- (C)1-C7) -alkyl, heteroarylcarbonyl- (C) 1-C7) -alkyl, heterocyclylcarbonyl- (C)1-C7) -alkyl, or
When Q represents Q-13, Q-14, Q-15, Q-25 and Q-26, R4And R5Together with the nitrogen or carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 membersOptionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R6represents hydrogen or (C)1-C7) -an alkyl group,
R8represents hydrogen, halogen, cyano, nitro, mercapto, hydroxy, NR10R11、OR12、SR13、SOR13、SO2R13Thiocyanato, isothiocyanato, formyl, (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyl, (C)2-C7) -alkynyl, (C)1-C8) -haloalkyl, (C)2-C7) -haloalkenyl, (C)2-C7) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) Halocycloalkenyl, pentafluorothio, (C)1-C7) -alkoxy- (C)1-C7) -haloalkyl, (C)1-C7) -haloalkoxy- (C)1-C7) -haloalkyl, (C)1-C7) -haloalkoxy- (C)1-C7) Alkyl, aryl- (C)1-C7) Alkyl, heteroaryl- (C)1-C7) Alkyl radicals, (C)3-C7) -cycloalkyl- (C)1-C7) Alkyl radicals, (C)4-C8) -cycloalkenyl- (C)1-C7) Alkyl, heterocyclyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkoxy- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylthio- (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkylthio- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylcarbonyl- (C) 1-C7) Alkyl, C (O) OR12、C(O)NR10R11、C(O)R12、-C＝NOR12、-C＝NOH、R10R11N-(C1-C7) -alkyl, R12O(O)C-(C1-C7) Alkyl, hydroxycarbonyl- (C)1-C7) Alkyl, aryl- (C)1-C7) -alkynyl, heteroaryl- (C)1-C7) -alkynyl, heterocyclyl- (C)1-C7) -alkynyl, tris [ (C)1-C7) -alkyl radical]Silyl radical- (C)2-C7) -alkynyl, bis [ (C)1-C7) -alkyl radical](aryl) silyl- (C)2-C7) -alkynyl, diaryl [ (C)1-C7) -alkyl radical]Silyl radical- (C)2-C7) -alkynyl, (C)3-C7) -cycloalkyl- (C)2-C7) -alkynyl, aryl- (C)2-C7) -alkenyl, heteroaryl- (C)2-C7) -alkenyl, heterocyclyl- (C)2-C7) -alkenyl, (C)3-C7) -cycloalkyl- (C)2-C7) -alkenyl, (C)1-C7) -alkoxy- (C)1-C7) -alkoxy- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylaminosulfonamido, (C)3-C7) -cycloalkylaminosulfonylamino, diazo, aryldiazo, tris [ (C)1-C7) -alkyl radical]Silyl, bis [ (C)1-C7) -alkyl radical](aryl) silyl, diaryl [ (C)1-C7) -alkyl radical]A silyl group (a) having a silyl group (a),
R10and R11Are identical or different and independently of one another represent hydrogen, (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyl, (C)2-C7) -alkynyl, (C)1-C7) Cyanoalkyl, (C)1-C8) -haloalkyl, (C)2-C7) -haloalkenyl, (C)2-C7) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) -halocycloalkenyl radical, (C)1-C7) -alkoxy- (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkoxy- (C)1-C7) Alkyl radicals, (C)1-C7) -alkylthio- (C)1-C7) Alkyl radicals, (C)1-C7) -haloalkylthio- (C) 1-C7) Alkyl radicals, (C)1-C7) -alkoxy- (C)1-C7) Haloalkyl, aryl- (C)1-C7) Alkyl, heteroaryl- (C)1-C7) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C7) Alkyl radicals, (C)4-C8) -cycloalkenyl- (C)1-C7) Alkyl radical, COR12、SO2R13、(C1-C7) -alkyl-HNO2S-、(C3-C8) -cycloalkyl-HNO2S-, heterocyclic group, (C)1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl radicals, (C)1-C7) Alkoxycarbonyl, aryl- (C)1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl, aryl- (C)1-C7) Alkoxycarbonyl, heteroaryl- (C)1-C7) Alkoxycarbonyl, (C)2-C7) -alkenyloxycarbonyl, (C)2-C7) -alkynyloxycarbonyl, heterocyclyl- (C)1-C7) -an alkyl group,
R12is represented by (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyl, (C)2-C7) -alkynyl, (C)1-C7) Cyanoalkyl, (C)1-C8) -haloalkyl, (C)2-C7) -haloalkenyl, (C)2-C7) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) -halocycloalkenyl radical, (C)1-C7) -alkoxy- (C)1-C7) Alkyl radicals, (C)1-C7) -alkoxy- (C)1-C7) Haloalkyl, aryl- (C)1-C7) Alkyl, heteroaryl- (C)1-C7) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C7) -alkyl radical、(C4-C8) -cycloalkenyl- (C)1-C7) Alkyl radicals, (C)1-C7) -alkoxycarbonyl- (C)1-C7) Alkyl radicals, (C)2-C7) -alkenyloxycarbonyl- (C)1-C7) Alkyl, aryl- (C)1-C7) -alkoxycarbonyl- (C)1-C7) -alkyl, hydroxycarbonyl- (C)1-C7) Alkyl, heterocyclyl- (C)1-C7) -an alkyl group,
R13is represented by (C) 1-C7) Alkyl radicals, (C)2-C7) -alkenyl, (C)2-C7) -alkynyl, (C)1-C7) Cyanoalkyl, (C)1-C8) -haloalkyl, (C)2-C7) -haloalkenyl, (C)2-C7) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) -halocycloalkenyl radical, (C)1-C7) -alkoxy- (C)1-C7) Alkyl radicals, (C)1-C7) -alkoxy- (C)1-C7) Haloalkyl, aryl- (C)1-C7) Alkyl, heteroaryl- (C)1-C7) Alkyl, heterocyclyl- (C)1-C7) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C7) Alkyl radicals, (C)4-C8) -cycloalkenyl- (C)1-C7) Alkyl, NR10R11，
R14And R15Independently of one another, represents hydrogen, (C)1-C7) -alkyl, halogen, or
R9And R15Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
and
w represents oxygen.
3. A compound of the general formula (I) and/or a salt thereof as claimed in claim 1, characterized in that
Q represents a group Q-1 to Q-30
Wherein the arrows represent the bond of the respective Q group to the nitrogen of the tetrahydropyrimidinone of the general formula (I),
A1、A2、A3、A4identical or different and, independently of one another, represent N (nitrogen) or a moiety C-R8But no more than two adjacent nitrogen atoms and according to the definition below, wherein the moiety C-R 8R of (A) to (B)8In each case having the same or different meanings, or
A1And A2When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A2And A3When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A3And A4When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted,
R1represents hydrogen, hydroxy, (C)1-C6) Alkyl radicals, (C)1-C6) -haloalkyl, (C)1-C6) -hydroxyalkyl, hydroxycarbonyl- (C)1-C6) Alkylene group, (C)1-C6) -alkoxy, (C)1-C6) -alkoxy- (C)1-C6) Alkylene group, (C)1-C6) Alkoxy-alkoxy (C)1-C6) -haloalkoxy, (C)3-C8) -cycloalkyl, (C)3-C8) Halocycloalkyl, aryl, heteroaryl, (C) 3-C8) -cycloalkyl- (C)1-C6) Alkylene, heterocyclic, (C)2-C6) -alkenyl, (C)2-C6) -alkenyloxy, (C)2-C6) -alkynyl, (C)2-C6) -alkynyloxy, amino, bis [ (C)1-C6) -alkyl radical]Amino, aryl- (C)1-C6) Alkylene, heteroaryl- (C)1-C6) Alkylene, heterocyclyl- (C)1-C6) Alkylene group, (C)1-C6) Cyanoalkyl, C (O) R12、C(O)OR12、C(O)NR10R11、SO2R13、R12O(O)C-(C1-C6) Alkylene, arylcarbonyl- (C)1-C6) Alkylene group, (C)1-C6) -alkylcarbonyl- (C)1-C6) Alkylene, heteroarylcarbonyl- (C)1-C6) Alkylene, heterocyclylcarbonyl- (C)1-C6) Alkylene group, (C)1-C6) -alkylcarbonyloxy- (C)1-C6) -an alkylene group,
R2and R9Independently of one another, represents hydrogen, hydroxy, fluorine, (C)1-C6) Alkyl radicals, (C)1-C6) -haloalkyl, (C)3-C8) Cycloalkyl, aryl, heteroaryl, heterocyclyl, aryl- (C)1-C6) -alkyl, heteroaryl- (C)1-C6) Alkyl, heterocyclyl- (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyl, (C)2-C6) -alkynyl, (C)1-C6) -alkoxy- (C)1-C6) -alkyl radical、(C1-C6) -haloalkoxy- (C)1-C6) Alkyl, aryl- (C)1-C6) -alkoxy- (C)1-C6) -alkyl, heteroaryl- (C)1-C6) -alkoxy- (C)1-C6) -alkyl, OR12、SR13、SOR13、SO2R13、NR10R11、R10R11N-(C1-C6) -alkyl, cyano- (C)1-C6) Alkyl, cyano, hydroxy- (C)1-C6) -alkyl, or
R1And R2Together with the nitrogen or carbon atom to which they are respectively attached form a fully or partially saturated ring having a total of 3 to 7 members, said ring being optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted, or
R2And R9Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R3represents hydroxy, mercapto, halogen, NR10R11、(C1-C6) -alkoxy, (C)3-C8) -cycloalkyl- (C)1-C6) Alkoxy, aryl- (C)1-C6) -alkoxy, (C)1-C6) -alkoxy- (C)1-C6) -alkoxy, arylcarbonyloxy, (C)1-C6) -alkylcarbonyloxy, (C)1-C6) -alkoxy- (C)1-C6) -alkylcarbonyloxy, aryl- (C)1-C6) -alkylcarbonyloxy, heteroarylcarbonyloxy, (C)3-C8) -cycloalkylcarbonyloxy, heterocyclylcarbonyloxy, (C)1-C6) -haloalkylcarbonyloxy, (C)2-C6) Alkenylcarbonyloxy, OC (O) OR12、OC(O)SR13、OC(S)OR12、OC(S)SR13、OSO2R13、OCHO，
R4And R7Independently of one another, represents hydrogen, mercapto, hydroxy, halogen, (C)1-C6) Alkyl radicals, (C)1-C6) -haloalkyl, (C)3-C8) -cycloalkyl, (C)3-C8) -cycloalkyl- (C)1-C6) Alkyl, aryl, heteroaryl, heterocyclyl, aryl- (C)1-C6) -alkyl, heteroaryl- (C)1-C6) Alkyl, heterocyclyl- (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyl, (C)2-C6) -alkynyl, (C)2-C6) -haloalkenyl, (C)2-C6) -haloalkynyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) Halocycloalkenyl, aryl- (C)2-C6) -alkenyl, heteroaryl- (C) 2-C6) -alkenyl, heterocyclyl- (C)2-C6) -alkenyl, aryl- (C)2-C6) -alkynyl, heteroaryl- (C)2-C6) -alkynyl, heterocyclyl- (C)2-C6) -alkynyl, (C)3-C8) -cycloalkyl- (C)2-C6) -alkynyl, arylcarbonyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylcarbonyl- (C)1-C6) -alkyl, heteroarylcarbonyl- (C)1-C6) Alkyl radicals, (C)3-C8) -cycloalkylcarbonyl- (C)1-C6) Alkyl, aryl- (C)1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkoxy- (C)1-C6) Alkyl, arylcarbonyloxy- (C)1-C6) Alkyl, heteroarylcarbonyloxy- (C)1-C6) Alkyl, heterocyclylcarbonyloxy- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylcarbonyloxy- (C)1-C6) Alkyl radicals, (C)3-C6) -cycloalkylcarbonyloxy- (C)1-C6) Alkyl radicals, (C)1-C6) -haloalkoxy- (C)1-C6) Alkyl, aryl- (C)1-C6) -alkoxy- (C)1-C6) -alkyl, heteroaryl- (C)1-C6) -alkoxy- (C)1-C6) Alkyl, CHO, C (O) R12、C(O)OR12、C(O)NR10R11、OR12、SR13、SOR13、SO2R13、NR10R11、R10R11N-(C1-C6) -alkyl, cyano- (C)1-C6) -alkyl, hydroxycarbonyl- (C)1-C6) -alkyl, hydroxycarbonyl, (C)1-C6) -haloalkoxy- (C)1-C6) Alkylthio group(s), (C)1-C6) -alkylthio- (C)1-C6) Alkylene group, (C)1-C6) -haloalkylthio- (C)1-C6) Alkylthio group(s), (C)1-C6) -alkylthio- (C)1-C6) Alkylthio, aminocarbonyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylaminocarbonyl- (C)1-C6) Alkyl radicals, (C)3-C6) -cycloalkylaminocarbonyl- (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyloxycarbonyl- (C) 1-C6) Alkyl radicals, (C)3-C6) -cycloalkyl- (C)1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl, cyano, hydroxy- (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyloxy- (C)1-C6) -alkyl, or
When Q represents Q-3, Q-4, Q-8, Q-9, Q-12, Q-13, Q-19 and Q-30, R4And R7Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R5represents hydrogen, formyl or (C)1-C6) -alkanesBase, (C)1-C6) Haloalkyl, hydroxy- (C)1-C6) -alkyl, hydroxycarbonyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkoxy- (C)1-C6) Alkyl radicals, (C)3-C8) -cycloalkyl, (C)3-C8) Halocycloalkyl, aryl, heteroaryl, (C)3-C8) -cycloalkyl- (C)1-C6) Alkyl, heterocyclyl, (C)2-C6) -alkenyl, (C)2-C6) -alkynyl, NR10R11Aryl group- (C)1-C6) -alkyl, heteroaryl- (C)1-C6) Alkyl, heterocyclyl- (C)1-C6) Alkyl radicals, (C)1-C6) Cyanoalkyl, C (O) R12、C(O)OR12、C(O)NR10R11、SO2R13、(C1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyloxycarbonyl- (C)1-C6) Alkyl, aryl- (C)1-C6) -alkoxycarbonyl- (C)1-C6) -alkyl, heteroaryl- (C)1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl, aryloxy carbonyl- (C)1-C6) -alkyl, arylcarbonyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylcarbonyl- (C)1-C6) -alkyl, heteroarylcarbonyl- (C) 1-C6) -alkyl, heterocyclylcarbonyl- (C)1-C6) -alkyl, or
When Q represents Q-13, Q-14, Q-15, Q-25 and Q-26, R4And R5Together with the nitrogen or carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R6represents hydrogen or (C)1-C6) -an alkyl group,
R8represents hydrogen, halogen, cyano, nitro, mercapto, hydroxy, NR10R11、OR12、SR13、SOR13、SO2R13Thiocyanato, isothiocyanato, formyl, (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyl, (C)2-C6) -alkynyl, (C)1-C8) -haloalkyl, (C)2-C6) -haloalkenyl, (C)2-C6) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) Halocycloalkenyl, pentafluorothio, (C)1-C6) -alkoxy- (C)1-C6) -haloalkyl, (C)1-C6) -haloalkoxy- (C)1-C6) -haloalkyl, (C)1-C6) -haloalkoxy- (C)1-C6) Alkyl, aryl- (C)1-C6) Alkyl, heteroaryl- (C)1-C6) Alkyl radicals, (C)3-C6) -cycloalkyl- (C)1-C6) Alkyl radicals, (C)4-C8) -cycloalkenyl- (C)1-C6) Alkyl, heterocyclyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkoxy- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylthio- (C)1-C6) Alkyl radicals, (C)1-C6) -haloalkylthio- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylcarbonyl- (C) 1-C6) Alkyl, C (O) OR12、C(O)NR10R11、C(O)R12、-C＝NOR12、-C＝NOH、R10R11N-(C1-C6) -alkyl, R12O(O)C-(C1-C6) Alkyl, hydroxycarbonyl- (C)1-C6) Alkyl, aryl- (C)1-C6) -alkynyl, heteroaryl- (C)1-C6) -alkynyl, heterocyclyl- (C)1-C6) -alkynyl, tris [ (C)1-C6) -alkyl radical]Silyl radical- (C)2-C6) -alkynyl, bis [ (C)1-C6) -alkyl radical](aryl) silyl- (C)2-C6) -alkynyl, diaryl [ (C)1-C6) -alkyl radical]Silyl radical- (C)2-C6) -alkynyl, (C)3-C6) -cycloalkyl- (C)2-C6) -alkynyl, aryl- (C)2-C6) -alkenyl, heteroaryl- (C)2-C6) -alkenyl, heterocyclyl- (C)2-C6) -alkenyl, (C)3-C6) -cycloalkyl- (C)2-C6) -alkenyl, (C)1-C6) -alkoxy- (C)1-C6) -alkoxy- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylaminosulfonamido, (C)3-C6) -cycloalkylaminosulfonylamino, diazo, aryldiazo, tris [ (C)1-C6) -alkyl radical]Silyl, bis [ (C)1-C6) -alkyl radical](aryl) silyl, diaryl [ (C)1-C6) -alkyl radical]A silyl group (a) having a silyl group (a),
R10and R11Are identical or different and independently of one another represent hydrogen, (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyl, (C)2-C6) -alkynyl, (C)1-C6) Cyanoalkyl, (C)1-C8) -haloalkyl, (C)2-C6) -haloalkenyl, (C)2-C6) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) -halocycloalkenyl radical, (C)1-C6) -alkoxy- (C)1-C6) Alkyl radicals, (C)1-C6) -haloalkoxy- (C)1-C6) Alkyl radicals, (C)1-C6) -alkylthio- (C)1-C6) Alkyl radicals, (C)1-C6) -haloalkylthio- (C) 1-C6) Alkyl radicals, (C)1-C6) -alkoxy- (C)1-C6) Haloalkyl, aryl- (C)1-C6) Alkyl, heteroaryl- (C)1-C6) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C6) Alkyl radicals, (C)4-C8) -cycloalkenyl- (C)1-C6) Alkyl radical, COR12、SO2R13、(C1-C6) -alkyl-HNO2S-、(C3-C8) -cycloalkyl-HNO2S-, heterocyclic group, (C)1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl radicals, (C)1-C6) Alkoxycarbonyl, aryl- (C)1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl, aryl- (C)1-C6) Alkoxycarbonyl, heteroaryl- (C)1-C6) Alkoxycarbonyl, (C)2-C6) -alkenyloxycarbonyl, (C)2-C6) -alkynyloxycarbonyl, heterocyclyl- (C)1-C6) -an alkyl group,
R12is represented by (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyl, (C)2-C6) -alkynyl, (C)1-C6) Cyanoalkyl, (C)1-C8) -haloalkyl, (C)2-C6) -haloalkenyl, (C)2-C6) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) -halocycloalkenyl radical, (C)1-C6) -alkoxy- (C)1-C6) Alkyl radicals, (C)1-C6) -alkoxy- (C)1-C6) Haloalkyl, aryl- (C)1-C6) Alkyl, heteroaryl- (C)1-C6) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C6) Alkyl radicals, (C)4-C8) -cycloalkenyl- (C)1-C6) Alkyl radicals, (C)1-C6) -alkoxycarbonyl- (C)1-C6) Alkyl radicals, (C)2-C6) -alkenyloxycarbonyl- (C)1-C6) Alkyl, aryl- (C)1-C6) -alkoxycarbonyl group-(C1-C6) -alkyl, hydroxycarbonyl- (C)1-C6) Alkyl, heterocyclyl- (C)1-C6) -an alkyl group,
R13is represented by (C) 1-C6) Alkyl radicals, (C)2-C6) -alkenyl, (C)2-C6) -alkynyl, (C)1-C6) Cyanoalkyl, (C)1-C8) -haloalkyl, (C)2-C6) -haloalkenyl, (C)2-C6) -haloalkynyl, (C)3-C8) -cycloalkyl, (C)3-C8) -halocycloalkyl, (C)4-C8) Cycloalkenyl radical, (C)4-C8) -halocycloalkenyl radical, (C)1-C6) -alkoxy- (C)1-C6) Alkyl radicals, (C)1-C6) -alkoxy- (C)1-C6) Haloalkyl, aryl- (C)1-C6) Alkyl, heteroaryl- (C)1-C6) Alkyl, heterocyclyl- (C)1-C6) Alkyl radicals, (C)3-C8) -cycloalkyl- (C)1-C6) Alkyl radicals, (C)4-C8) -cycloalkenyl- (C)1-C6) Alkyl, NR10R11，
R14And R15Independently of one another, represents hydrogen, (C)1-C6) -alkyl, fluoro, or
R9And R15Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
and
w represents oxygen.
4. A compound of the general formula (I) and/or a salt thereof as claimed in claim 1, characterized in that
Q represents a group Q-1 to Q-30
Wherein the arrows represent the bond of the respective Q group to the nitrogen of the tetrahydropyrimidinone of the general formula (I),
A1、A2、A3、A4identical or different and, independently of one another, represent N (nitrogen) or a moiety C-R8But no more than two adjacent nitrogen atoms and according to the definition above, wherein part of C-R 8R of (A) to (B)8In each case having the same or different meanings, or
A1And A2When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A2And A3When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted, or
A3And A4When each is a group C-R8When taken together with the atoms to which they are attached form a fully saturated, partially saturated or fully unsaturated 5 to 7 membered ring, optionally interrupted by a heteroatom selected from N, O and S, and optionally further substituted,
R1represents hydrogen, methyl, ethyl, n-propyl, 1-methylethyl, n-butyl, 1-methylprop-1-yl, 2-methylprop-1-yl, 1-dimethylethyl-1-yl, n-pentyl, 1-methylbut-1-yl, 2-methylbut-1-yl, 3-methylbut-1-yl, 1-dimethylprop-1-yl, 1, 2-dimethylprop-1-yl, 2-dimethylprop-1-yl, 1-ethylprop-1-yl, n-hexyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1-methylethyl, n-butyl, 1-methylprop-1-yl, 1- -dimethylbutyl, 1, 2-dimethylbutyl, 1, 3-dimethylbutyl, 2, 2-dimethylbutyl, 2, 3-dimethylbutyl, 3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1, 2-trimethylpropyl, 1,2, 2-trimethylpropyl, 1-ethyl-1-methylpropyl, 1-ethyl-2-methylpropyl, trifluoromethyl, pentafluoroethyl, 1,2, 2-tetrafluoroethyl, heptafluoro-n-propyl, heptafluoroisopropyl, nonafluorobutyl, chlorodifluoromethyl, bromodifluoromethyl, dichlorofluoromethyl, iododifluoromethyl, bromofluoromethyl, 1-fluoroethyl, 2-fluoroethyl, fluoromethyl, difluoromethyl, 2, 2-difluoroethyl, 2, 2-dimethylpropyl, 1-ethylpropyl, 1-ethylmethyl, 2-difluoroethyl, 2,2,2, 2-trifluoroethyl, 3,3, 3-trifluoroprop-1-yl, 3,3, 3-trifluoroprop-2-yl, difluoro-tert-butyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, spiro [2.2]Pent-1-yl, spiro [2.3 ]]Hex-1-yl, spiro [2.3 ]]Hex-4-yl, 3-spiro [2.3 ]]Hex-5-yl, spiro [3.3 ]]Hept-1-yl, spiro [3.3 ]]Hept-2-yl, bicyclo [1.1.0]But-1-yl, bicyclo [1.1.0]But-2-yl, bicyclo [2.1.0]Pent-1-yl, bicyclo [1.1.1]Pent-1-yl, bicyclo [2.1.0]Pent-2-yl, bicyclo [2.1.0]Pentan-5-yl, bicyclo [2.1.1]Hexyl, bicyclo [2.2.1]Hept-2-yl, bicyclo [2.2.2]Oct-2-yl, adamantan-1-yl, adamantan-2-yl, 1-methylcyclopropyl, 2-dimethylcyclopropyl, 2, 3-dimethylcyclopropyl, 1 '-bis (cyclopropyl) -1-yl, 1' -bis (cyclopropyl) -2-yl, 2 '-methyl-1, 1' -bis (cyclopropyl) -2-yl, 1-cyanocyclopropyl, 2-cyanocyclopropyl, 1-methylcyclobutyl, 2-methylcyclobutyl, 3-methylcyclobutyl, 1-cyanocyclobutyl, 2-cyanocyclobutyl, 3-cyanocyclobutyl, 1-allylcyclopropyl, 1-vinylcyclobutyl, 2-cyanocyclobutyl, 1-allylcyclopropyl, 2-vinylcyclobutyl, 2-methylcyclobutyl, etc, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 1-methoxycyclohexyl, 2-methoxycyclohexyl, 3-methoxycyclohexyl, cyclopropylmethyl, cyclobutylmethyl, cyclopentylmethyl, cyclohexylmethyl, phenyl, p-F-phenyl, m-F-phenyl, o-F-phenyl, p-Cl-phenyl, m-Cl-phenyl, o-Cl-phenyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, thiophen-2-yl, thiophen-3-yl, furan-2-yl, methyl ethyl, propyl, butyl, furan-3-yl, tetrahydrofuran-2-yl, tetrahydrofuran-3-yl, benzyl, p-Cl-benzyl, p-F-benzyl, p-methoxybenzyl, p-methylbenzyl, p-trifluoromethyl Benzyl, p-nitrobenzyl, m-Cl-benzyl, m-F-benzyl, m-methoxybenzyl, m-methylbenzyl, o-Cl-benzyl, o-F-benzyl, o-methoxybenzyl, o-methylbenzyl, 1-phenyleth-1-yl, 2-phenyleth-1-yl, 1- (o-chlorophenyl) eth-1-yl, 1- (o-fluorophenyl) eth-1-yl, 1- (o-methylphenyl) eth-1-yl, 1- (o-bromophenyl) eth-1-yl, 1- (o-iodophenyl) eth-1-yl, pyridin-2-ylmethyl, pyridin-3-ylmethyl, pyridin-4-ylmethyl, pyrimidin-2-ylmethyl, m-methoxybenzyl, m-methylbenzyl, o-Cl-benzyl, o-F-, Pyrimidin-4-ylmethyl, tetrahydrofuran-2-ylmethyl, o-cyanophenylmethyl, m-cyanophenylmethyl, p-cyanophenylmethyl, cyanomethyl, cyanoethyl, methoxycarbonyl, ethoxycarbonyl, n-propoxycarbonyl, isopropoxycarbonyl, t-butoxycarbonyl, benzyloxycarbonyl, allyloxycarbonyl, methylcarbonyl, ethylcarbonyl, n-propylcarbonyl, isopropylcarbonyl, n-butylcarbonyl, 1-methylprop-1-ylcarbonyl, 2-methylprop-1-ylcarbonyl, 1-dimethyleth-1-ylcarbonyl, phenylcarbonyl, methylaminocarbonyl, dimethylaminocarbonyl, ethylaminocarbonyl, n-propylaminocarbonyl, isopropylaminocarbonyl, n-butylaminocarbonyl, t-butylaminocarbonyl, benzylaminocarbonyl, p-cyanophenylmethyl, cyanomethyl, n-propylcarbonyl, 1-methylprop-1-ylcarbonyl, 2-methylprop-1-, Methoxycarbonylmethyl, ethoxycarbonylmethyl, tert-butoxycarbonylmethyl, benzyloxycarbonylmethyl, methoxycarbonylethyl, ethoxycarbonylethyl, tert-butoxycarbonylmethyl, benzyloxycarbonylmethyl, methylcarbonyloxymethyl, ethylcarbonyloxymethyl, n-propylcarbonyloxymethyl, 1-methylethylcarbonyloxymethyl, 1-dimethylethylcarbonyloxymethyl, hydroxycarbonylmethyl, hydroxycarbonylethyl, hydroxycarbonyln-propyl, methoxy, ethoxy, n-propoxy, isopropoxy, methoxymethyl, ethoxymethyl, n-propoxymethyl, isopropoxymethyl, n-butoxymethyl, methoxyethyl, ethoxyethyl, n-propoxyethyl, isopropoxyethyl, methoxy-n-propyl, ethoxy-n-propyl, methoxy-n-butyl, amino, dimethylamino, methyl (ethyl) amino, methyl, n-propyl, n, Diethylamino, cyanomethyl, cyanoethyl, prop-2-yn-1-yl,
R2And R9Independently of one another, represents hydrogen, hydroxy, fluorine, methyl, ethyl, n-propyl-yl, isopropyl, n-butyl, 1-methylpropan-1-yl, 2-methylpropan-1-yl, 1-dimethylethyl-1-yl, trifluoromethyl, difluoromethyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, phenyl, p-F-phenyl, m-F-phenyl, o-F-phenyl, p-Cl-phenyl, m-Cl-phenyl, o-Cl-phenyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, thiophen-2-yl, thiophen-3-yl, furan-2-yl, furan-3-yl, methoxymethyl, methoxy-1-yl, 2-methylpropan-1-yl, 1-dimethylethyl-1-yl, p-Cl-phenyl, m-Cl-phenyl, o-Cl-phenyl, pyridin-2-yl, pyridin, Ethoxymethyl, methoxyethyl, ethoxyethyl, methoxy, ethoxy, n-propoxy, isopropoxy, trifluoromethoxy, difluoromethoxy, methylthio, ethylthio, trifluoromethylthio, dimethylamino, methylamino, diethylamino, methyl (ethyl) amino, cyano, or
R1And R2Together with the nitrogen or carbon atom to which they are respectively attached form a fully or partially saturated ring having a total of 3 to 7 members, said ring being optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted, or
R2And R9Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R3Represents hydroxy, mercapto, fluoro, chloro, bromo, iodo, methoxy, ethoxy, n-propoxy, 1-methylethoxy, n-butoxy, 1-methylpropoxy, 2-methylpropoxy, 1-dimethylethoxy, n-pentyloxy, 1-methylbutoxy, 2-methylbutoxy, 3-methylbutoxy, 1-dimethylpropoxy, 1, 2-dimethylpropoxy, 2-dimethylpropoxy, 1-ethylpropoxy, n-hexyloxy, 1-methylpentyloxy, 2-methylpentyloxy, 3-methylpentyloxy, 4-methylpentyloxy, 1-dimethylbutyloxy, 1, 2-dimethylbutyloxy, 1, 3-dimethylbutyloxy, 2-dimethylbutyloxy, n-butyloxy, 1-methylpropyloxy, 2-methylbutoxy, 3-methylbutoxy, 2, 3-dimethylbutoxy, 3-dimethylbutoxy, 1-ethylbutoxy, 2-ethylbutoxy, 1, 2-trimethylpropoxy, 1,2, 2-trimethylpropoxy, 1-ethyl-1-methylpropoxy, 1-ethan-e2-methylpropyloxy, cyclopropylmethoxy, cyclobutylmethoxy, cyclopentylmethoxy, cyclohexylmethoxy, benzyloxy, p-chlorophenylmethoxy, m-chlorophenylmethoxy, o-chlorophenylmethoxy, p-methoxyphenylmethoxy, p-nitrophenylmethoxy, methoxymethoxy, methoxyethoxy, methoxy-n-propoxy, methoxy-n-butoxy, ethoxymethoxy, ethoxyethoxy, ethoxy-n-propoxy, ethoxy-n-butoxy, n-propoxymethoxy, isopropoxymethoxy, methylcarbonyloxy, ethylcarbonyloxy, n-propylcarbonyloxy, 1-methylethylcarbonyloxy, n-butylcarbonyloxy, 1-methylpropylcarbonyloxy, 2-methylpropylcarbonyloxy, 1-dimethylethylcarbonyloxy, n-pentylcarbonyloxy, p-chlorophenylmethoxy, p-nitrophenylmethyloxy, m-n-propylcarbonyloxy, 1-methylbutylcarbonyloxy, 2-methylbutylcarbonyloxy, 3-methylbutylcarbonyloxy, 1-dimethylpropylcarbonyloxy, 1, 2-dimethylpropylcarbonyloxy, 2-dimethylpropylcarbonyloxy, 1-ethylpropylcarbonyloxy, n-hexylcarbonyloxy, 1-methylpentylcarbonyloxy, 2-methylpentylcarbonyloxy, 3-methylpentylcarbonyloxy, 4-methylpentylcarbonyloxy, 1-dimethylbutylcarbonyloxy, 1, 2-dimethylbutylcarbonyloxy, 1, 3-dimethylbutylcarbonyloxy, 2-dimethylbutylcarbonyloxy, 2, 3-dimethylbutylcarbonyloxy, 3-dimethylbutylcarbonyloxy, 1-ethylbutylcarbonyloxy, 2-methylpentylcarbonyloxy, 2, 3-dimethylbutylcarbonyloxy, 2, 3-dimethylbutylcarbonyloxy, 3-, 2-ethylbutylcarbonyloxy, 1, 2-trimethylpropylcarbonyloxy, 1,2, 2-trimethylpropylcarbonyloxy, 1-ethyl-1-methylpropylcarbonyloxy, 1-ethyl-2-methylpropylcarbonyloxy, phenylcarbonyloxy, p-chlorophenylcarbonyloxy, m-chlorophenylcarbonyloxy, o-chlorophenylcarbonyloxy, p-fluorophenylcarbonyloxy, m-fluorophenylcarbonyloxy, o-fluorophenylcarbonyloxy, benzylcarbonyloxy, thien-2-ylcarbonyloxy, furan-2-ylcarbonyloxy, cyclopropylcarbonyloxy, cyclobutylcarbonyloxy, cyclopentylcarbonyloxy, cyclohexylcarbonyloxy, 1-fluorocycloprop-1-ylcarbonyloxy, 1-chlorocycloprop-1-ylcarbonyloxy, 1-chloroprop-1-ylcarbonyloxy, 1-cyanocyclopropyl1-ylcarbonyloxy, 1-methylcyclopropyl1-ylcarbonyloxy, 1-trifluoromethylcyclopropyl1-ylcarbonyloxy, adamantylcarbonyloxy, trifluoromethyl Carbonyloxy, difluoromethylcarbonyloxy, methoxycarbonyloxy, ethoxycarbonyloxy, n-propoxycarbonyloxy, isopropoxycarbonyloxy, n-butoxycarbonyloxy, 1-dimethylethoxycarbonyl-oxy, 2-dimethylpropoxycarbonyloxy, benzyloxycarbonyloxy, allyloxycarbonyloxy, cyclopropyloxycarbonyloxy, cyclobutoxycarbonyloxy, cyclopentyloxycarbonyloxy, cyclohexyloxycarbonyloxy, cyclopropylmethoxycarbonyloxy, cyclobutylmethoxycarbonyloxy, cyclopentylmethoxycarbonyloxy, cyclohexylmethoxycarbonyloxy, 3,3, 3-trifluoroethoxycarbonyloxy, 2-difluoroethoxycarbonyloxy, pyridin-2-ylcarbonyloxy, pyridin-3-ylcarbonyloxy, pyridin-4-ylcarbonyloxy, n-propoxycarbonyloxy, n-butyloxycarbonyloxy, 1-dimethylethoxycarbonyl-2, 2-dimethylpropoxycarbonyloxy, 4-trifluoromethylpyridin-3-ylcarbonyloxy, allylcarbonyloxy, methylsulfonyloxy, ethylsulfonyloxy, n-propylsulfonyloxy, 1-methylethylsulfonyloxy, cyclopropylsulfonyloxy, cyclobutylsulfonyloxy, cyclopentylsulfonyloxy, cyclohexylsulfonyloxy, phenylsulfonyloxy, p-chlorophenylsulfonyloxy, m-chlorophenylsulfonyloxy, o-chlorophenylsulfonyloxy, p-fluorophenylsulfonyloxy, m-fluorophenylsulfonyloxy, o-fluorophenylsulfonyloxy, p-methoxyphenylsulfonyloxy, m-methoxyphenylsulfonyloxy, o-methoxyphenylsulfonyloxy, p-methylphenylsulfonyloxy, m-methylphenylsulfonyloxy, o-methylphenylsulfonyloxy,
R4And R7Independently of one another, represents hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, mercapto, methyl, ethyl, n-propyl, 1-methylethyl, n-butyl, 1-methylpropyl, 2-methylpropyl, 1-dimethylethyl, n-pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 1-dimethylpropyl, 1, 2-dimethylpropyl, 2-dimethylpropyl, 1-ethylpropyl, n-hexyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1-dimethylbutyl, 1, 2-dimethylbutyl, 1, 3-dimethylbutyl, 2-dimethylbutyl, 2, 3-dimethylbutyl, 3-dimethylbutyl, methyl-butyl, ethyl-1, 2-dimethylbutyl, 1-methylethyl, 2-methylbutyl, 2-methylpropyl, 2-dimethylbutyl, 3, 1-ethylbutyl, 2-ethylbutyl, 1, 2-trimethylpropyl, 1,2, 2-trimethylpropyl, 1-ethyl-1-methylpropyl, 1-ethyl-2-methylPropyl, trifluoromethyl, pentafluoroethyl, 1,2, 2-tetrafluoroethyl, heptafluoro-n-propyl, heptafluoro-isopropyl, nonafluorobutyl, chlorodifluoromethyl, bromodifluoromethyl, dichlorofluoromethyl, iododifluoromethyl, bromofluoromethyl, 1-fluoroethyl, 2-fluoroethyl, fluoromethyl, difluoromethyl, 2, 2-difluoroethyl, 2,2, 2-trifluoroethyl, difluorotert-butyl, chloromethyl, bromomethyl, fluoromethyl, 3,3, 3-trifluoro-n-propyl, 1-fluoroprop-1-yl, 1-trifluoromethylprop-1-yl, 2-trifluoromethylprop-2-yl, 1-fluoroprop-1-yl, 2-fluoroprop-2-yl, 2-chloroprop-2-yl, cyclopropyl, cyclobutyl, cyclopropyl, heptafluoroisopropyl, nonafluorobutyl, chlorodifluoromethyl, chloromethyl, bromomethyl, 3, 3-trifluoro-n-propyl, 1-fluoroprop-1-yl, 1-fluoroprop-2-yl, cyclopentyl, cyclohexyl, 1-methylcycloprop-1-yl, 2-dimethylcycloprop-1-yl, 2, 3-dimethylcyclopropyl, 1-cyanocycloprop-1-yl, 2-cyanocycloprop-1-yl, 1-methylcyclobutyl, 2-methylcyclobutyl, 3-dimethylcyclobutyl, 1-cyanocyclobutyl, 2-cyanocyclobutyl, 3-cyanocyclobutyl, 1-allylcyclopropyl, 1-vinylcyclobutyl, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 1-methoxycyclohexyl, 2-methylcycloprop-1-yl, 2-cyanocycloprophenyl, 1-ethylcyclobutyl, 1-vinylcyclobutyl, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 1-methoxycyclohexyl, 2-methoxycyclohexyl, 3-methoxycyclohexyl, spiro [2.2 ] ]Pent-1-yl, spiro [2.3 ]]Hex-1-yl, spiro [2.3 ]]Hex-4-yl, 3-spiro [2.3 ]]Hex-5-yl, spiro [3.3 ]]Hept-1-yl, spiro [3.3 ]]Hept-2-yl, bicyclo [1.1.0]But-1-yl, bicyclo [1.1.0]But-2-yl, bicyclo [2.1.0]Pent-1-yl, bicyclo [1.1.1]Pent-1-yl, bicyclo [2.1.0]Pent-2-yl, bicyclo [2.1.0]Pentan-5-yl, bicyclo [2.1.1]Hexyl, bicyclo [2.2.1]Hept-2-yl, bicyclo [2.2.2]Oct-2-yl, bicyclo [3.2.1]Oct-2-yl, bicyclo [3.2.2]Non-2-yl group, adamantan-1-yl group, adamantan-2-yl group, cyclopropylmethyl group, cyclobutylmethyl group, cyclopentylmethyl group, cyclohexylmethyl group, phenyl group, 2-fluorophenyl group, 3-fluorophenyl group, 4-fluorophenyl group, 2, 4-difluorophenyl group, 2, 5-difluorophenyl group, 2, 6-difluorophenyl group, 2, 3-difluorophenyl group, 3, 4-difluorophenyl group, 3, 5-difluorophenyl group, 2,4, 5-trifluorophenyl group, 3,4, 5-trifluorophenyl group, 2-chlorophenyl group, 3-chlorophenyl group, 4-chlorophenyl group, 2, 4-dichlorophenyl group, 2, 5-dichlorophenyl group, 2, 6-dichlorophenyl group, 2, 3-dichlorophenyl group, 3, 4-dichlorophenyl group, 3, 5-dichlorophenyl group, 2,4, 5-trichlorophenyl group, 3,4, 5-trichlorophenyl group, 2,4, 6-trichlorophenyl group, 2-bromophenyl group, 3-bromophenyl group, 4-bromophenyl group, 2-iodophenyl group, 3-iodophenyl group, 4-iodophenyl groupIodophenyl, 2-bromo-4-fluorophenyl, 2-bromo-4-chlorophenyl, 3-bromo-4-fluorophenyl, 3-bromo-4-chlorophenyl, 3-bromo-5-fluorophenyl, 3-bromo-5-chlorophenyl, 2-fluoro-4-bromophenyl, 2-chloro-4-bromophenyl, 3-fluoro-4-bromophenyl, 3-chloro-4-bromophenyl, 2-chloro-4-fluorophenyl, 3-chloro-4-fluorophenyl, 2-fluoro-3-chlorophenyl, 2-fluoro-4-chlorophenyl, 2-fluoro-5-chlorophenyl, 3-fluoro-4-chlorophenyl, 3-fluoro-5-chlorophenyl group, 2-fluoro-6-chlorophenyl group, 2-methylphenyl group, 3-methylphenyl group, 4-methylphenyl group, 2, 4-dimethylphenyl group, 2, 5-dimethylphenyl group, 2, 6-dimethylphenyl group, 2, 3-dimethylphenyl group, 3, 4-dimethylphenyl group, 3, 5-dimethylphenyl group, 2,4, 5-trimethylphenyl group, 3,4, 5-trimethylphenyl group, 2,4, 6-trimethylphenyl group, 2-methoxyphenyl group, 3-methoxyphenyl group, 4-methoxyphenyl group, 2, 4-dimethoxyphenyl group, 2, 5-dimethoxyphenyl group, 2, 6-dimethoxyphenyl group, 2, 3-dimethoxyphenyl group, 3, 4-dimethoxyphenyl group, 3, 5-dimethoxyphenyl group, 2,4, 5-trimethoxyphenyl group, 3,4, 5-trimethoxyphenyl group, 2,4, 6-trimethoxyphenyl group, 2-trifluoromethoxyphenyl group, 3-trifluoromethoxyphenyl group, 4-trifluoromethoxyphenyl group, 2-difluoromethoxyphenyl group, 3-difluoromethoxyphenyl group, 4-difluoromethoxyphenyl group, 2-trifluoromethylphenyl group, 3-trifluoromethylphenyl group, 4-trifluoromethylphenyl group, 2-difluoromethylphenyl group, 3-difluoromethylphenyl group, 4-difluoromethylphenyl group, 3, 5-bis (trifluoromethyl) phenyl group, 3-trifluoromethyl-5-fluorophenyl group, 3-trifluoromethyl-5-chlorophenyl group, 2-trifluoromethyl-5-fluorophenyl group, and 3-trifluoromethyl-5-chlorophenyl group, 3-methyl-5-fluorophenyl group, 3-methyl-5-chlorophenyl group, 3-methoxy-5-fluorophenyl group, 3-methoxy-5-chlorophenyl group, 3-trifluoromethoxy-5-chlorophenyl group, 2-ethoxyphenyl group, 3-ethoxyphenyl group, 4-ethoxyphenyl group, 2-methylthiophenyl group, 3-methylthiophenyl group, 4-methylthiophenyl group, 2-trifluoromethylthienyl group, 3-trifluoromethylthienyl group, 4-trifluoromethylthienyl group, 2-ethylphenyl group, 3-ethylphenyl group, 4-ethylphenyl group, 2-methoxycarbonylphenyl group, 3-methoxycarbonylphenyl group, 4-methoxycarbonylphenyl group, 2-ethoxycarbonylphenyl group, 3-ethoxycarbonylphenyl group, 2-ethoxycarbonylphenyl group, 3-ethoxyphenyl group, 2-ethoxy, 3-ethoxycarbonylphenyl, 4-ethoxycarbonylphenyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrazin-2-yl, pyridazin-3-yl, pyridazin-4-yl, pyrimidin-2-yl, pyrimidin-5-yl, pyrimidin-4-yl, pyridazin-3-ylmethyl, pyridazin-4-ylmethyl, pyrimidin-2-ylmethyl, pyrimidin-5-ylmethyl Yl, pyrimidin-4-ylmethyl, pyrazin-2-ylmethyl, 3-chloropyrazin-2-yl, 3-bromopyrazin-2-yl, 3-methoxypyrazin-2-yl, 3-ethoxypyrazin-2-yl, 3-trifluoromethylpyrazin-2-yl, 3-cyanopyrazin-2-yl, naphthalen-1-yl, quinolin-4-yl, quinolin-6-yl, quinolin-8-yl, quinolin-2-yl, quinoxalin-2-yl, 2-naphthylmethyl, 1-naphthylmethyl, quinolin-4-ylmethyl, quinolin-6-ylmethyl, quinolin-8-ylmethyl, pyrazin-2-ylmethyl, 3-chloropyrazin-2-yl, 3-cyanopyrazin-2-yl, and/or benzyl, Quinolin-2-ylmethyl, quinoxalin-2-ylmethyl, pyrazin-2-ylmethyl, 4-chloropyridin-2-yl, 3-chloropyridin-4-yl, 2-chloropyridin-3-yl, 2-chloropyridin-4-yl, 2-chloropyridin-5-yl, 2, 6-dichloropyridin-4-yl, 3-chloropyridin-5-yl, 3, 5-dichloropyridin-2-yl, 3-chloro-5-trifluoromethylpyridin-2-yl, (4-chloropyridin-2-yl) methyl, (3-chloropyridin-4-yl) methyl, (2-chloropyridin-3-yl) methyl, (2-chloropyridin-4-yl) methyl, (2-chloropyridin-5-yl) methyl, (2, 6-dichloropyridin-4-yl) methyl, (3-chloropyridin-5-yl) methyl, (3, 5-dichloropyridin-2-yl) methyl, thiophen-2-yl, thiophen-3-yl, 5-methylthion-2-yl, 5-ethylthiophen-2-yl, 5-chlorothien-2-yl, 5-bromothiophen-2-yl, 4-methylthiophen-2-yl, 3-methylthiophen-2-yl, 5-fluorothiophen-3-yl, 3, 5-dimethylthiophen-2-yl, methyl-thiophen-2-yl, methyl, 3-ethylthiophen-2-yl, 4, 5-dimethylthiophen-2-yl, 3, 4-dimethylthiophen-2-yl, 4-chlorothien-2-yl, furan-2-yl, 5-methylfuran-2-yl, 5-ethylfuran-2-yl, 5-methoxycarbonylfuran-2-yl, 5-chlorofuran-2-yl, 5-bromofuran-2-yl, thien-3-yl, sulfolane-2-yl, sulfolane-3-yl, tetrahydrothiopyran-4-yl, tetrahydropyran-4-yl, tetrahydrofuran-2-yl, tetrahydrothiopyran-2-yl, 5-methylfuran-2-yl, 5-ethylfuran-2-yl, 5-methoxycarbonylfuran-2-yl, 5-chlorothiofuran-, Tetrahydrofuran-3-yl, 1- (4-methylphenyl) ethyl, 1- (3-methylphenyl) ethyl, 1- (2-methylphenyl) ethyl, 1- (4-chlorophenyl) ethyl, 1- (3-chlorophenyl) ethyl, 1- (2-chlorophenyl) ethyl, benzyl, (4-fluorophenyl) methyl, (3-fluorophenyl) methyl, (2, 4-difluorophenyl) methyl, (3, 5-difluorophenyl) methyl, (2, 6-difluorophenyl) methyl, (2,4, 5-trifluorophenyl) methyl, (2,4, 6-trifluorophenyl) methyl, (4-chlorophenyl) methyl, 1- (4-methylphenyl) ethyl, 1- (2-fluorophenyl) methyl, 3-fluorophenyl) methyl, 2-fluorophenyl) methyl, 5-difluorophenyl) methyl, 2,4, (3-chlorophenyl) methyl group, (2, 4-dichlorophenyl) methyl group, (3, 5-dichlorophenyl) methyl group, (2, 5-dichlorophenyl) methyl group, and (2, 6-dichlorobenzene) Phenyl) methyl group, (2,4, 5-trichlorophenyl) methyl group, (2,4, 6-trichlorophenyl) methyl group, (4-bromophenyl) methyl group, (3-bromophenyl) methyl group, (2-bromophenyl) methyl group, (4-iodophenyl) methyl group, (3-iodophenyl) methyl group, (2-iodophenyl) methyl group, (3-chloro-5-trifluoromethylpyridin-2-yl) methyl group, (2-bromo-4-fluorophenyl) methyl group, (2-bromo-4-chlorophenyl) methyl group, (3-bromo-4-fluorophenyl) methyl group, (3-bromo-4-chlorophenyl) methyl group, (3-bromo-5-fluorophenyl) methyl group, (3-bromo-5-chlorophenyl) methyl group, (2-fluoro-4-bromophenyl) methyl group, (2-chloro-4-bromophenyl) methyl group, (3-fluoro-4-bromophenyl) methyl group, (3-chloro-4-bromophenyl) methyl group, (2-chloro-4-fluorophenyl) methyl group, (3-chloro-4-fluorophenyl) methyl group, (2-fluoro-3-chlorophenyl) methyl group, (2-fluoro-4-chlorophenyl) methyl group, (2-fluoro-5-chlorophenyl) methyl group, (3-fluoro-4-chlorophenyl) methyl group, (3-fluoro-5-chlorophenyl) methyl group, (2-fluoro-6-chlorophenyl) methyl group, 2-phenyleth-1-yl group, 3-trifluoromethyl-4-chlorophenyl group, methyl group, phenyl group, 3-chloro-4-trifluoromethylphenyl group, 2-chloro-4-trifluoromethylphenyl group, 3, 5-difluoropyridin-2-yl group, (3, 6-dichloropyridin-2-yl) methyl group, (4-trifluoromethylphenyl) methyl group, (3-trifluoromethylphenyl) methyl group, (2-trifluoromethylphenyl) methyl group, (4-trifluoromethoxyphenyl) methyl group, (3-trifluoromethoxyphenyl) methyl group, (2-trifluoromethoxyphenyl) methyl group, (4-methoxyphenyl) methyl group, (3-methoxyphenyl) methyl group, (2-methoxyphenyl) methyl group, (4-methylphenyl) methyl group, (3-methylphenyl) methyl group, (2-methylphenyl) methyl group, (4-cyanophenyl) methyl group, phenyl group, (3-cyanophenyl) methyl, (2, 4-diethylphenyl) methyl, (3, 5-diethylphenyl) methyl, (3, 4-dimethylphenyl) methyl, (3, 5-dimethoxyphenyl) methyl, 1-phenyleth-1-yl, 1- (o-chlorophenyl) eth-1-yl, 1, 3-thiazol-2-yl, 4-methyl-1, 3-thiazol-2-yl, vinyl, 1-propenyl, 2-propenyl, 1-methylvinyl, 1-butenyl, 2-butenyl, 3-butenyl, 1-methyl-1-propenyl, 1-methyl-1-butenyl, 2-butenyl, 3-butenyl, 1-methyl-1-propenyl, methyl-1-ethyl-1-methyl-ethyl, 2-methyl-1-propenyl, 1-methyl-2-propenyl, 2-methyl-2-propenyl, 1-pentenyl, 2-pentenyl, 3-pentenyl, 4-pentenyl, 1-methyl-1-butenyl, 2-methyl-1-butenyl, 3-methyl-1-butenyl, 1-methyl-2-butenyl, 2-methyl-2-butenyl, 3-methyl-2-butenyl, 1-methyl-3-butenyl, 2-methyl-3-butenyl, 3-methyl-3-butenyl, 1-dimethyl-1-butenyl A group-2-propenyl group, a 1, 2-dimethyl-1-propenyl group, a 1, 2-dimethyl-2-propenyl group, a 1-ethyl-1-propenyl group, a 1-ethyl-2-propenyl group, a 1-hexenyl group, a 2-hexenyl group, a 3-hexenyl group, a 4-hexenyl group, a 5-hexenyl group, a 1-methyl-1-pentenyl group, a 2-methyl-1-pentenyl group, a 3-methyl-1-pentenyl group, a 4-methyl-1-pentenyl group, a 1-methyl-2-pentenyl group, a 2-methyl-2-pentenyl group, a 3-methyl-2-pentenyl group, a 4-methyl-2-pentenyl group, a, 1-methyl-3-pentenyl, 2-methyl-3-pentenyl, 3-methyl-3-pentenyl, 4-methyl-3-pentenyl, 1-methyl-4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4-pentenyl, 1-dimethyl-2-butenyl, 1-dimethyl-3-butenyl, 1, 2-dimethyl-1-butenyl, 1, 2-dimethyl-2-butenyl, 1, 2-dimethyl-3-butenyl, 1, 3-dimethyl-1-butenyl, 1, 3-two methyl 2-butene radical, 1, 3-two methyl 3-butene radical, 2-two methyl 3-butene radical, 2, 3-two methyl 1-butene radical, 2, 3-two methyl 2-butene radical, 2, 3-two methyl 3-butene radical, 3-two methyl 1-butene radical, 3-two methyl 2-butene radical, 1-ethyl-1-butene radical, 1-ethyl-2-butene radical, 1-ethyl-3-butene radical, 2-ethyl-1-butene radical, 2-ethyl-2-butene radical, 2-ethyl-3-butene radical, 2-ethyl-1-butene radical, 1,1, 2-trimethyl-2-propenyl, 1-ethyl-1-methyl-2-propenyl, 1-ethyl-2-methyl-1-propenyl and 1-ethyl-2-methyl-2-propenyl, ethynyl, 1-propynyl, 2-propynyl, 1-butynyl, 2-butynyl, 3-butynyl, 1-methyl-2-propynyl, 1-pentynyl, 2-pentynyl, 3-pentynyl, 4-pentynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl, 2-methyl-3-butynyl, 3-methyl-1-butynyl, 1-ethyl-2-propenyl, 1-ethyl-1-methyl-butynyl, 1-ethyl-2-propynyl, 1-methyl-2-butynyl, 1,1, 1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 1-hexynyl, 2-hexynyl, 3-difluorocyclobut-1-yl, 3-fluorocyclobut-1-yl, 1-fluorocyclobut-1-yl, 2-difluorocycloprop-1-yl, 1-fluorocycloprop-1-yl, 2-fluorocycloprop-1-yl, 4-fluorocyclohexyl, 4-difluorocyclohexyl, methoxycarbonylmethyl, ethoxycarbonylmethyl, n-propoxycarbonylmethyl, isopropoxycarbonylmethyl, n-butoxycarbonylmethyl, tert-butoxycarbonylmethyl, methoxymethyl, ethoxymethyl, n-propoxymethyl, isopropoxymethyl, N-butoxymethyl, methoxyethyl, ethoxyethyl, n-propoxyethyl, isopropoxy Phenylethyl group, methoxy-n-propyl group, methoxy-n-butyl group, trifluoromethoxy-methyl group, difluoromethoxymethyl group, 2, 2-difluoroethoxymethyl group, 2,2, 2-trifluoroethoxymethyl group, trifluoromethoxyethyl group, difluoromethoxyethyl group, 2, 2-difluoroethoxyethyl group, 2,2, 2-trifluoroethoxyethyl group, methoxycarbonyl group, ethoxycarbonyl group, n-propoxycarbonyl group, isopropoxycarbonyl group, n-butoxycarbonyl group, t-butoxycarbonyl group, allyloxycarbonyl group, benzyloxycarbonyl group, methylcarbonyl group, ethylcarbonyl group, n-propylcarbonyl group, isopropylcarbonyl group, n-butylcarbonyl group, t-butylcarbonyl group, phenylcarbonyl group, p-chlorophenylcarbonyl group, m-chlorophenylcarbonyl group, o-chlorophenylcarbonyl group, p-fluorophenylcarbonyl group, m-fluorophenylcarbonyl group, o-fluorophenylcarbonyl group, p-methoxyphenylcarbonyl group, m, O-methoxyphenylcarbonyl, p-trifluoromethylphenylcarbonyl, m-trifluoromethylphenylcarbonyl, o-trifluoromethylphenylcarbonyl, methoxy, ethoxy, n-propoxy, isopropoxy, benzyloxy, p-chlorophenylmethoxy, phenoxy, p-chlorophenoxy, m-chlorophenoxy, o-chlorophenoxy, p-fluorophenoxy, m-fluorophenoxy, o-fluorophenoxy, p-methoxyphenoxy, m-methoxyphenoxy, o-methoxyphenoxy, p-trifluoromethylphenoxy, m-trifluoromethylphenoxy, o-trifluoromethylphenoxy, methylaminocarbonyl, ethylaminocarbonyl, n-propylaminocarbonyl, isopropylaminocarbonyl, cyclopropylaminocarbonyl, cyclobutylaminocarbonyl, cyclopentylaminocarbonyl, cyclohexylaminocarbonyl, cyclopropylmethylaminocarbonyl, cyclobutylmethylaminocarbonyl, cyclopentylmethylaminocarbonyl, cyclohexylmethylaminocarbonyl, Dimethylaminocarbonyl, diethylaminocarbonyl, benzylmethylaminocarbonyl, methylamino, dimethylamino, ethylamino, diethylamino, n-propylamino, isopropylamino, cyclopropylamino, cyclobutylamino, cyclopentylamino, cyclohexylamino, benzylamino, cyanomethyl, cyanoethyl, 3-cyanoprop-1-yl, 2-cyanoprop-1-yl, 1-cyanoprop-1-yl, 2-cyanoprop-2-yl, 2-cyano-1, 1-dimethyleth-1-yl, 1- (cyanomethyl) -1-methylprop-1-yl, hydroxycarbonyl, hydroxycarbonylmethyl, hydroxycarbonylethyl, CHO, methoxyethylthio, ethoxyethylethylethylthio, ethoxyethylthio Thio, trifluoromethoxy ethylthio, pentafluoroethoxyethylthio, methylthioethylthio, ethylthioethylthio, trifluoromethylthioethylthio, pentafluorothioethylthio, benzylthio, p-chlorophenyl-methylthio, m-chlorophenyl-methylthio, o-chlorophenyl-methylthio, p-fluorophenyl-methylthio, m-fluorophenyl-methylthio, o-fluorophenyl-methylthio, ethylthio, n-propylthio, i-propylthio, n-butylthio, t-butylthio, cyclobutylthio, cyclopentylthio, cyclohexylthio, phenylthio, pyridin-2-ylthio, pyridin-3-ylthio, pyridin-4-ylthio, p-chlorophenylthio, m-chlorophenylthio, o-chlorophenylthio, p-fluorophenylthio, m-fluorophenylthio, o-fluorophenylthio, p-methoxyphenylthio, m-methoxyphenylthio, o-methylphenylthio, p-methylphenylthio, M-methylphenylsulfanyl, o-methylphenylsulfanyl, methylsulfonyl, ethylsulfonyl, n-propylsulfonyl, 1-methylethylsulfonyl, cyclopropylsulfonyl, cyclobutylsulfonyl, cyclopentylsulfonyl, cyclohexylsulfonyl, phenylsulfonyloxy, p-chlorophenylsulfonyl, m-chlorophenylsulfonyl, o-chlorophenylsulfonyl, p-fluorophenylsulfonyl, m-fluorophenylsulfonyl, o-fluorophenylsulfonyl, p-methoxyphenylsulfonyl, m-methoxyphenylsulfonyl, o-methoxyphenylsulfonyl, p-methylphenylsulfonyl, m-methylphenylsulfonyl, o-methylphenylsulfonyl, 2-methoxyprop-2-yl, 2-ethoxyprop-2-yl, 2-n-propoxyprop-2-yl, 2-n-butoxyprop-2-yl, 2-benzyloxyprop-2-yl, 2-Phenylethoxypropan-2-yl, 2-trifluoromethoxypropan-2-yl, 2-difluoromethoxypropan-2-yl, 2,2, 2-trifluoroethoxypropan-2-yl, 2, 2-difluoroethoxypropan-2-yl, 2- (4-chlorophenylmethoxy) propan-2-yl, 2- (4-fluorophenylmethoxy) propan-2-yl, 2- (4-bromophenylmethoxy) propan-2-yl, 2- (4-trifluoromethylphenylmethoxy) propan-2-yl, 2- (4-methylphenylmethoxy) propan-2-yl, 2- (3-chlorophenylmethoxy) propan-2-yl, methyl-ethyl-2-yl, methyl-2-propyl-2-yl, methyl-propyl-2-yl, 2- (3-fluorophenylmethoxy) propan-2-yl, 2- (3-bromophenylmethoxy) propan-2-yl, 2- (3-trifluoromethylphenylmethoxy) propan-2-yl, 2- (3-methylphenylmethoxy) propan-2-yl, 2- (2-chlorophenylmethoxy) propan-2-yl, 2- (2-fluorophenylmethoxy) propan-2-yl, 2- (2-bromophenylmethoxy) propan-2-yl, 2- (2-trifluoromethylphenylmethoxy) propan-2-yl Methoxy) prop-2-yl, 2- (2-methylphenylmethoxy) prop-2-yl, 2- (methoxymethyl) prop-2-yl, 2- (ethoxymethyl) prop-2-yl, 2-methoxycarbonylprop-2-yl, 2-ethoxycarbonylprop-2-yl, 2-hydroxycarbonylprop-2-yl, 2-aminocarbonylprop-2-yl, aminocarbonyl, aminocarbonylmethyl, aminocarbonylethyl, cyano, hydroxymethyl, hydroxyethyl, 2-hydroxyprop-2-yl, allyloxymethyl, 2-allyloxyethyl, 2-allyloxypropyl-2-yl, or
When Q represents Q-3, Q-4, Q-8, Q-9, Q-12, Q-13, Q-19 and Q-30, R4And R7Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R5represents hydrogen, formyl, methyl, ethyl, n-propyl, 1-methylethyl, n-butyl, 1-methylpropyl, 2-methylpropyl, 1-dimethylethyl, n-pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, 1-dimethylpropyl, 1, 2-dimethylpropyl, 2-dimethylpropyl, 1-ethylpropyl, n-hexyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1-dimethylbutyl, 1, 2-dimethylbutyl, 1, 3-dimethylbutyl, 2-dimethylbutyl, 2, 3-dimethylbutyl, 3-dimethylbutyl, 1-ethylbutyl, n-butyl, 1-methylpropyl, 2-dimethylpropyl, 2-dimethylpropyl, 1-ethylpropyl, 1-dimethylpropyl, 1-methylpentyl, 2, 2-ethylbutyl group, 1, 2-trimethylpropyl group, 1,2, 2-trimethylpropyl group, 1-ethyl-1-methylpropyl group, 1-ethyl-2-methylpropyl group, 2, 2-difluoroethyl group, 2,2, 2-trifluoroethyl group, 3,3, 3-trifluoro-n-propyl group, methoxymethyl group, ethoxymethyl group, methoxyethyl group, ethoxyethyl group, methoxy-n-propyl group, methoxy-n-butyl group, ethoxy-n-propyl group, ethoxy-n-butyl group, hydroxyethyl group, hydroxy-n-propyl group, hydroxycarbonylmethyl group, hydroxycarbonylethyl group, hydroxycarbonyln-propyl group, methoxycarbonylmethyl group, ethoxycarbonylmethyl group, n-propoxycarbonylmethyl group, isopropoxycarbonylmethyl group, t-butoxycarbonylmethyl group, methoxycarbonylethyl group, ethoxycarbonylethyl group, n-propoxycarbonylethyl group, Isopropoxycarbonylethyl, tert-butoxycarbonylethyl, methoxycarbonyl-n-propyl, ethoxycarbonyl N-propyl, benzyloxycarbonylmethyl, benzyloxycarbonylethyl, allyloxycarbonylmethyl, allyloxycarbonylethyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, 1-methylcycloprop-1-yl, 2-dimethylcycloprop-1-yl, 2, 3-dimethylcyclopropyl, 1-cyanopropyl, 2-cyanopropyl, 1-methylcyclobutyl, 2-methylcyclobutyl, 3-dimethylcyclobutyl, 1-cyanocyclobutyl, 2-cyanocyclobutyl, 3-cyanocyclobutyl, 1-allylcyclopropyl, 1-vinylcyclobutyl, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, cyclohexylmethyl, propylmethyl, 1-methylcyclopropyl, 2-cyanocyclobutyl, 1-cyanopropyl, 2-cyanocyclobutyl, 2-methylcyclohexyl group, 3-methylcyclohexyl group, 1-methoxycyclohexyl group, 2-methoxycyclohexyl group, 3-methoxycyclohexyl group, cyclopropylmethyl group, cyclobutylmethyl group, cyclopentylmethyl group, cyclohexylmethyl group, cyanomethyl group, 2-cyanoeth-1-yl group, 1-cyanoeth-1-yl group, cyano-n-propyl group, methoxycarbonyl group, ethoxycarbonyl group, t-butoxycarbonyl group, benzyloxycarbonyl group, n-butoxycarbonyl group, allyloxycarbonyl group, methylcarbonyl group, ethylcarbonyl group, n-propylcarbonyl group, isopropylcarbonyl group, n-butylcarbonyl group, t-butylcarbonyl group, phenylcarbonyl group, p-chlorophenylcarbonyl group, m-chlorophenylcarbonyl group, o-chlorophenylcarbonyl group, p-fluorophenylcarbonyl group, m-fluorophenylcarbonyl group, o-fluorophenylcarbonyl group, p-methoxyphenylcarbonyl group, m-, O-methoxyphenylcarbonyl, p-trifluoromethylphenylcarbonyl, m-trifluoromethylphenylcarbonyl, o-trifluoromethylphenylcarbonyl, methylaminocarbonyl, ethylaminocarbonyl, isopropylaminocarbonyl, n-propylaminocarbonyl, phenylaminocarbonyl, p-Cl-phenylaminocarbonyl, m-Cl-phenylaminocarbonyl, o-Cl-phenylaminocarbonyl, cyclopropylaminocarbonyl, cyclobutylaminocarbonyl, cyclopentylaminocarbonyl, cyclohexylaminocarbonyl, cyclopropylmethylaminocarbonyl, cyclobutylmethylaminocarbonyl, cyclopentylmethylaminocarbonyl, cyclohexylmethylaminocarbonyl, dimethylaminocarbonyl, diethylaminocarbonyl, benzyl (methyl) aminocarbonyl, prop-2-en-1-yl, prop-2-yn-1-yl, 1-fluorocycloprop-1-yl, di-n-propylmethyl-aminocarbonyl, di-n-butylaminocarbonyl, di-methyl-phenylaminocarbonyl, di-l-2-en-1-yl, di-, 2-fluoropropn-1-yl group, 2-difluorocycloprop-1-yl group, 3-difluorocyclobutane-1-yl group, phenyl group, 2-fluorophenyl group, 3-fluorophenyl group, 4-fluorophenyl group, 2, 4-difluorophenyl group, 2, 5-difluorophenyl group, 2, 6-difluorophenyl group Phenyl, 2, 3-difluorophenyl, 3, 4-difluorophenyl, 3, 5-difluorophenyl, 2,4, 5-trifluorophenyl, 3,4, 5-trifluorophenyl, 2-chlorophenyl, 3-chlorophenyl, 4-chlorophenyl, 2, 4-dichlorophenyl, 2, 5-dichlorophenyl, 2, 6-dichlorophenyl, 2, 3-dichlorophenyl, 3, 4-dichlorophenyl, 3, 5-dichlorophenyl, 2,4, 5-trichlorophenyl, 3,4, 5-trichlorophenyl, 2,4, 6-trichlorophenyl, 2-bromophenyl, 3-bromophenyl, 4-bromophenyl, 2-iodophenyl, 3-iodophenyl, 4-iodophenyl, 2-bromo-4-fluorophenyl, 2-bromo-4-chlorophenyl, 3-bromo-4-fluorophenyl, 3-bromo-4-chlorophenyl, 3-bromo-5-fluorophenyl, 3-bromo-5-chlorophenyl, 2-fluoro-4-bromophenyl, 2-chloro-4-bromophenyl, 3-fluoro-4-bromophenyl, 3-chloro-4-bromophenyl, 2-chloro-4-fluorophenyl, 3-chloro-4-fluorophenyl, 2-fluoro-3-chlorophenyl, 2-fluoro-4-chlorophenyl, 2-fluoro-5-chlorophenyl, 3-fluoro-4-chlorophenyl, 3-fluoro-5-chlorophenyl, 2-fluoro-6-chlorophenyl, 2-methylphenyl, 2-bromo-4-chlorophenyl, 3-bromo-5-fluorophenyl, 3-chloro-4-bromophenyl, 2-chloro-4-chlorophenyl, 2-fluoro-6-chlorophenyl, 2-methylphenyl, 3-methylphenyl, 4-methylphenyl, 2, 4-dimethylphenyl, 2, 5-dimethylphenyl, 2, 6-dimethylphenyl, 2, 3-dimethylphenyl, 3, 4-dimethylphenyl, 3, 5-dimethylphenyl, 2,4, 5-trimethylphenyl, 3,4, 5-trimethylphenyl, 2,4, 6-trimethylphenyl, 2-methoxyphenyl, 3-methoxyphenyl, 4-methoxyphenyl, 2, 4-dimethoxyphenyl, 2, 5-dimethoxyphenyl, 2, 6-dimethoxyphenyl, 2, 3-dimethoxyphenyl, 3, 4-dimethoxyphenyl, 3, 5-dimethoxyphenyl, 2,4, 5-trimethoxyphenyl, 3,4, 5-trimethoxyphenyl group, 2,4, 6-trimethoxyphenyl group, 2-trifluoromethoxyphenyl group, 3-trifluoromethoxyphenyl group, 4-trifluoromethoxyphenyl group, 2-difluoromethoxyphenyl group, 3-difluoromethoxyphenyl group, 4-difluoromethoxyphenyl group, 2-trifluoromethylphenyl group, 3-trifluoromethylphenyl group, 4-trifluoromethylphenyl group, 2-difluoromethylphenyl group, 3-difluoromethylphenyl group, 4-difluoromethylphenyl group, 3, 5-di (trifluoromethyl) phenyl group, 3-trifluoromethyl-5-fluorophenyl group, 3-trifluoromethyl-5-chlorophenyl group, 3-methyl-5-fluorophenyl group, 3-methyl-5-chlorophenyl group, 3-methoxy-5-fluorophenyl group, 2-trifluoromethoxyphenyl group, 3-trifluoromethyl-5-fluorophenyl group, and the like, 3-methoxy-5-chlorophenyl group, 3-trifluoromethoxy-5-chlorophenyl group, 2-ethoxyphenyl group, 3-ethoxyphenyl group, 4-ethoxyphenyl group, 2-methylthiophenyl group, 3-methylthiophenyl group, 4-methylthiophenyl group, 2-trifluoromethylthienyl group, 3-trifluoromethylthienyl group, 4-trifluoromethylthienyl group, methoxymethyl group, 2-ethylthio group, etc Alkylphenyl, 3-ethylphenyl, 4-ethylphenyl, 2-methoxycarbonylphenyl, 3-methoxycarbonylphenyl, 4-methoxycarbonylphenyl, 2-ethoxycarbonylphenyl, 3-ethoxycarbonylphenyl, 4-ethoxycarbonylphenyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrazin-2-yl, pyridazin-3-yl, pyridazin-4-yl, pyrimidin-2-yl, pyrimidin-5-yl, pyrimidin-4-yl, pyridazin-3-ylmethyl, pyridazin-4-ylmethyl, pyrimidin-2-ylmethyl, pyrimidin-5-ylmethyl, pyrimidin-4-ylmethyl, pyrazin-2-ylmethyl, pyrazin-4-ylmethyl, pyridazin-4-ylmethyl, and mixtures thereof, 3-chloropyrazin-2-yl, 3-bromopyrazin-2-yl, 3-methoxypyrazin-2-yl, 3-ethoxypyrazin-2-yl, 3-trifluoromethylpyrazin-2-yl, 3-cyanopyrazin-2-yl, naphthalen-1-yl, quinolin-4-yl, quinolin-6-yl, quinolin-8-yl, quinolin-2-yl, quinoxalin-2-yl, 2-naphthylmethyl, 1-naphthylmethyl, quinolin-4-ylmethyl, quinolin-6-ylmethyl, quinolin-8-ylmethyl, quinolin-2-ylmethyl, quinoxalin-2-ylmethyl, naphthalen-2-ylpyrazin-2-ylmethyl, naphthalen-2, Pyrazin-2-ylmethyl, 4-chloropyridin-2-yl, 3-chloropyridin-4-yl, 2-chloropyridin-3-yl, 2-chloropyridin-4-yl, 2-chloropyridin-5-yl, 2, 6-dichloropyridin-4-yl, 3-chloropyridin-5-yl, 3, 5-dichloropyridin-2-yl, 3-chloro-5-trifluoromethylpyridin-2-yl, (4-chloropyridin-2-yl) methyl, (3-chloropyridin-4-yl) methyl, (2-chloropyridin-3-yl) methyl, (2-chloropyridin-4-yl) methyl, (2-chloropyridin-5-yl) methyl, (2, 6-dichloropyridin-4-yl) methyl, (3-chloropyridin-5-yl) methyl, (3, 5-dichloropyridin-2-yl) methyl, thiophen-2-yl, thiophen-3-yl, 5-methylthion-2-yl, 5-ethylthiophen-2-yl, 5-chlorothien-2-yl, 5-bromothiophen-2-yl, 4-methylthion-2-yl, 3-methylthion-2-yl, 5-fluorothiophen-3-yl, 3, 5-dimethylthiophen-2-yl, 3-ethylthiophen-2-yl, 4, 5-dimethylthiophen-2-yl, 3-ethylthiophen-2-yl, 3-chloropyridin-2-yl, 5-bromothiophen-2-yl, 5-methylthion-2-yl, 3, 4-dimethylthiophen-2-yl, 4-chlorothien-2-yl, furan-2-yl, 5-methylfuran-2-yl, 5-ethylfuran-2-yl, 5-methoxycarbonylfuran-2-yl, 5-chlorofuran-2-yl, 5-bromofuran-2-yl, thien-3-yl, sulfolane-2-yl, sulfolane-3-yl, benzyl, (4-fluorophenyl) methyl, (3-fluorophenyl) methyl, (2, 4-difluorophenyl) methyl, (3, 5-difluorophenyl) methyl, (2, 5-difluorophenyl) methyl, methyl, (2, 6-difluorophenyl) methyl, (2,4, 5-trifluorophenyl) methyl, and (2,4, 6-trifluoro-phenyl) methyl Phenyl) methyl group, (4-chlorophenyl) methyl group, (3-chlorophenyl) methyl group, (2, 4-dichlorophenyl) methyl group, (3, 5-dichlorophenyl) methyl group, (2, 6-dichlorophenyl) methyl group, (2,4, 5-trichlorophenyl) methyl group, (2,4, 6-trichlorophenyl) methyl group, (4-bromophenyl) methyl group, (3-bromophenyl) methyl group, (2-bromophenyl) methyl group, (4-iodophenyl) methyl group, (3-iodophenyl) methyl group, (2-iodophenyl) methyl group, (3-chloro-5-trifluoromethylpyridin-2-yl) methyl group, (2-bromo-4-fluorophenyl) methyl group, methyl, (2-bromo-4-chlorophenyl) methyl group, (3-bromo-4-fluorophenyl) methyl group, (3-bromo-4-chlorophenyl) methyl group, (3-bromo-5-fluorophenyl) methyl group, (3-bromo-5-chlorophenyl) methyl group, (2-fluoro-4-bromophenyl) methyl group, (2-chloro-4-bromophenyl) methyl group, (3-fluoro-4-bromophenyl) methyl group, (3-chloro-4-bromophenyl) methyl group, (2-chloro-4-fluorophenyl) methyl group, (3-chloro-4-fluorophenyl) methyl group, (2-fluoro-3-chlorophenyl) methyl group, (2-fluoro-4-chlorophenyl) methyl group, (2-fluoro-5-chlorophenyl) methyl group, (3-fluoro-4-chlorophenyl) methyl group, (3-fluoro-5-chlorophenyl) methyl group, (2-fluoro-6-chlorophenyl) methyl group, phenethyl group, 3-trifluoromethyl-4-chlorophenyl group, 3-chloro-4-trifluoromethylphenyl group, 2-chloro-4-trifluoromethylphenyl group, 3, 5-difluoropyridin-2-yl group, (3, 6-dichloropyridin-2-yl) methyl group, (4-trifluoromethylphenyl) methyl group, (3-trifluoromethylphenyl) methyl group, (2-trifluoromethylphenyl) methyl group, (4-trifluoromethoxyphenyl) methyl group, (3-trifluoromethoxyphenyl) methyl group, benzyl, (2-trifluoromethoxyphenyl) methyl group, (4-methoxyphenyl) methyl group, (3-methoxyphenyl) methyl group, (2-methoxyphenyl) methyl group, (4-methylphenyl) methyl group, (3-methylphenyl) methyl group, (2-methylphenyl) methyl group, (4-cyanophenyl) methyl group, (3-cyanophenyl) methyl group, (2, 4-diethylphenyl) methyl group, (3, 5-diethylphenyl) methyl group, (3, 4-dimethylphenyl) methyl group, (3, 5-dimethoxyphenyl) methyl group, 1-phenyleth-1-yl group, methylsulfonyl group, ethylsulfonyl group, n-propylsulfonyl group, 1-methylethylsulfonyl group, cyclopropylsulfonyl group, cyclobutylsulfonyl group, butylsulfonyl group, isopropylsulfonyl group, and the like, Cyclopentylsulfonyl, cyclohexylsulfonyl, phenylsulfonyloxy, p-chlorophenylsulfonyl, m-chlorophenylsulfonyl, o-chlorophenylsulfonyl, p-fluorophenylsulfonyl, m-fluorophenylsulfonyl, o-fluorophenylsulfonyl, p-methoxyphenylsulfonyl, m-methoxyphenylsulfonyl, O-methoxyphenylsulfonyl, p-methylphenylsulfonyl, m-methylphenylsulfonyl, o-methylphenylsulfonyl, phenylcarbonylmethyl, p-chlorophenylcarbonylmethyl, m-chlorophenylcarbonylmethyl, o-chlorophenylcarbonylmethyl, p-fluorophenylcarbonylmethyl, m-fluorophenylcarbonylmethyl, o-fluorophenylcarbonylmethyl, methylcarbonylmethyl, ethylcarbonylmethyl, n-propylcarbonylmethyl, i-propylcarbonylmethyl, n-butylcarbonylmethyl, t-butylcarbonylmethyl, or
When Q represents Q-13, Q-14, Q-15, Q-25 and Q-26, R4And R5Together with the nitrogen or carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
R6represents hydrogen, methyl, ethyl, or a mixture thereof,
R8represents hydrogen, halogen, cyano, nitro, mercapto, hydroxy, methylamino, ethylamino, isopropylamino, N-propylamino, dimethylamino, diethylamino, cyclopropylamino, cyclobutylamino, cyclopentylamino, cyclohexylamino, methoxycarbonylmethylamino, methoxycarbonylethylamino, ethoxycarbonylmethylamino, ethoxycarbonylethylamino, methoxycarbonylamino, ethoxycarbonylamino, tert-butoxycarbonylamino, phenylamino, N-piperidinyl, N-pyrrolidinyl, N-morpholinyl, methylaminocarbonylamino, ethylaminocarbonylamino, N-propylaminocarbonylamino, isopropylaminocarbonylamino, benzylaminocarbonylamino, phenylaminocarbonylamino, p-Cl-phenylaminocarbonylamino, m-Cl-phenylaminocarbonylamino, methyl-amino, methylamino, N-propylamino, methoxycarbonylamino, ethoxycarbonylamino, N-propylamino, ethoxycarbonylamino, tert-butoxycarbonylamino, phenylamino, N-piperidinyl, N-pyrrolidinyl, N-morpholinyl, methylaminocarbonylamino, ethylaminocarbonylamino, N-propylamin, o-Cl-phenylaminocarbonylamino, cyclopropylaminocarbonylamino, cyclobutylaminocarbonylamino, cyclopentylaminocarbonylamino, cyclohexylaminocarbonylamino, dimethylaminocarbonylamino, methoxy, ethoxy, n-propoxy, isopropoxy, n-butoxy, tert-butoxy, methoxycarbonyloxy, ethoxycarbonyloxy, tert-butoxycarbonyloxy, methylaminocarbonyloxy, ethylaminocarbonyloxy, n-propylaminocarbonyloxy, cyclohexylaminocarbonylamino, methylaminocarbonyloxy, ethylaminocarbonyloxy, isopropylaminocarbonyloxy, cyclopentyloxycarbonyloxy, Isopropylaminocarbonyloxy, benzylaminocarbonyloxy, phenylaminocarbonyloxy, cyclopropylaminocarbonyloxy, cyclobutylaminocarbonyloxy, cyclopentylaminocarbonyloxy, cyclohexylaminocarbonyloxy, dimethylaminocarbonyloxy, phenoxy, p-Cl-phenoxy, o-Cl-phenoxy, m-trifluoromethylphenoxy, p-trifluoromethylphenoxy, trifluoromethoxy, difluoromethoxy, 2, 2-difluoroethoxy, 2,2, 2-trifluoroethoxy, methylthio, ethylthio, n-propylthio, isopropylthio, phenylthio, p-Cl-phenylthio, m-Cl-phenylthio, o-Cl-phenylthio, pyridin-2-ylthio, pyridin-3-ylthio, o-Cl-phenylthio, p-chloro-, Benzylthio, trifluoromethylthio, pentafluoroethylthio, cyclopropylthio, cyclobutylthio, cyclopentylthio, cyclohexylthio, methylsulfinyl, ethylsulfinyl, n-propylsulfinyl, isopropylsulfinyl, n-butylsulfinyl, tert-butylsulfinyl, phenylsulfinyl, benzylsulfinyl, pyridin-2-ylsulfinyl, methylsulfonyl, ethylsulfonyl, n-propylsulfonyl, isopropylsulfonyl, n-butylsulfonyl, tert-butylsulfonyl, phenylsulfonyl, benzylsulfonyl, pyridin-2-ylsulfonyl, methyl, ethyl, n-propyl, 1-methylethyl, n-butyl, 1-methylpropyl, 2-methylpropyl, 1-dimethylethyl, n-pentyl, 1-methylbutyl, 2-methylbutyl, 3-methylbutyl, butylthio, ethylthio, n-propylthio, phenylsulfonyl, benzylsulfonyl, isopropylsulfonyl, n-, 1, 1-dimethylpropyl, 1, 2-dimethylpropyl, 2, 2-dimethylpropyl, 1-ethylpropyl, n-hexyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1-dimethylbutyl, 1, 2-dimethylbutyl, 1, 3-dimethylbutyl, 2, 2-dimethylbutyl, 2, 3-dimethylbutyl, 3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1, 2-trimethylpropyl, 1,2, 2-trimethylpropyl, 1-ethyl-1-methylpropyl, 1-ethyl-2-methylpropyl, thiocyanato, isothiocyanato, formyl, vinyl, 1-propenyl, 2-propenyl, 1-methylethenyl, 1-butenyl, 2-butenyl, 3-butenyl, 1-methyl-1-propenyl, 2-methyl-1-propenyl, 1-methyl-2-propenyl, 2-methyl-2-propenyl, 1-pentenyl, 2-pentenyl, 3-pentenyl, 4-pentenyl, 1-methyl-1-butenyl, 2-methyl-1-butenyl, 3-methyl-1-butenyl -1-butenyl, 1-methyl-2-butenyl, 2-methyl-2-butenyl, 3-methyl-2-butenyl, 1-methyl-3-butenyl, 2-methyl-3-butenyl, 3-methyl-3-butenyl, 1-dimethyl-2-propenyl, 1, 2-dimethyl-1-propenyl, 1, 2-dimethyl-2-propenyl, 1-ethyl-1-propenyl, 1-ethyl-2-propenyl, ethynyl, 1-propynyl, 2-propynyl, 1-butynyl, 2-butynyl, 3-butynyl, 1-methyl-2-propynyl, 2-butynyl, 3-butynyl, 1-methyl-2-propynyl, and the like, 1-pentynyl, 2-pentynyl, 3-pentynyl, 4-pentynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl, 2-methyl-3-butynyl, 3-methyl-1-butynyl, 1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 1-hexynyl, 2-hexynyl, 3-difluorocyclobut-1-yl, 3-fluorocyclobut-1-yl, 1-fluorocyclobut-1-yl, 2-difluorocycloprop-1-yl, 1-fluorocycloprop-1-yl, 2-fluorocycloprop-1-yl, 1-fluorocycloprop-2-methylprop-1-yl, 4-fluorocyclohexyl, 4-difluorocyclohexyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, 1-methylcycloprop-1-yl, 2-dimethylcycloprop-1-yl, 2, 3-dimethylcyclopropyl, 1-cyanopropyl, 2-cyanopropyl, 1-methylcyclobutyl, 2-methylcyclobutyl, 3-dimethylcyclobutyl, 1-cyanocyclobutyl, 2-cyanocyclobutyl, 3-cyanocyclobutyl, 1-allylcyclopropyl, 1-vinylcyclobutyl, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-dimethylcyclohexyl, 1-vinylcyclopropyl, 2-cyanocyclopropyl, 1-allylcyclopropyl, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-butylcyclopropyl, 3-methylcyclohexyl, 1-methoxycyclohexyl, 2-methoxycyclohexyl, 3-methoxycyclohexyl, spiro [2.2 ] ]Pent-1-yl, spiro [2.3 ]]Hex-1-yl, spiro [2.3 ]]Hex-4-yl, 3-spiro [2.3 ]]Hex-5-yl, spiro [3.3 ]]Hept-1-yl, spiro [3.3 ]]Hept-2-yl, bicyclo [1.1.0]But-1-yl, bicyclo [1.1.0]But-2-yl, bicyclo [2.1.0]Pent-1-yl, bicyclo [1.1.1]Pent-1-yl, bicyclo [2.1.0]Pent-2-yl, bicyclo [2.1.0]Pentan-5-yl, bicyclo [2.1.1]Hexyl, bicyclo [2.2.1]Hept-2-yl, bicyclo [2.2.2]Oct-2-yl, bicyclo [3.2.1]Oct-2-yl, bicyclo [3.2.2]Nonan-2-yl, adamantan-1-yl, adamantan-2-yl, cyclopropylmethyl, cyclobutylmethyl, cyclopentylmethyl, cyclohexylmethyl, trifluoromethyl, pentafluoroethyl, 1,2, 2-tetrafluoroethyl, heptafluoro-n-propyl, heptafluoro-isopropyl, nonafluorobutyl, chlorodifluoromethyl, bromodifluoromethyl, dichlorofluoromethyl, iododifluoromethyl, bromofluoromethyl, 1-fluoroethyl,2-fluoroethyl, fluoromethyl, difluoromethyl, 2, 2-difluoroethyl, 2,2, 2-trifluoroethyl, difluoro-tert-butyl, chloromethyl, bromomethyl, fluoromethyl, 3,3, 3-trifluoro-n-propyl, methoxycarbonyl, ethoxycarbonyl, isopropoxycarbonyl, n-propoxycarbonyl, n-butoxycarbonyl, tert-butoxycarbonyl, benzyloxycarbonyl, allyloxycarbonyl, methylaminocarbonyl, ethylaminocarbonyl, n-propylaminocarbonyl, isopropylaminocarbonyl, benzylaminocarbonyl, phenylaminocarbonyl, cyclopropylaminocarbonyl, cyclobutylaminocarbonyl, cyclopentylaminocarbonyl, cyclohexylaminocarbonyl, dimethylaminocarbonyl, diethylaminocarbonyl, allylaminocarbonyl, pentafluorothio, methoxydifluoromethyl, ethoxydifluoromethyl, n-propoxydifluoromethyl, trifluoromethyl, Trifluoromethoxyethyl, trifluoromethoxy-n-propyl, methoxymethyl, ethoxymethyl, n-propoxymethyl, ethoxyethyl, methoxyethyl, n-propoxyethyl, methoxy-n-propyl, ethoxy-n-propyl, 1-methoxyethyl-1-yl, 1-methoxyprop-1-yl, 1-ethoxyeth-1-yl, 2-methoxyprop-2-yl, 2-ethoxyprop-2-yl, methylthiomethyl, methylthioethyl, methylthion-propyl, ethylthiomethyl, trifluoromethylthiomethyl, pentafluoroethylthiomethyl, trifluoromethylthioethyl, trifluoromethylthio-n-propyl, methylcarbonyl, ethylcarbonyl, isopropylcarbonyl, n-butylcarbonyl, tert-butylcarbonyl, phenylcarbonyl, o-Cl-phenylcarbonyl, o-propylcarbonyl, n-propyloxymethyl, 2-methoxypropyl, 2-ethoxypropyl, 2-ethylthiomethyl, methylthioethyl, m-Cl-phenylcarbonyl, p-Cl-phenylcarbonyl, methoxycarbonylmethyl, ethoxycarbonylmethyl, methoxycarbonylethyl, ethoxycarbonylethyl, n-propoxycarbonylmethyl, t-butoxycarbonylmethyl, t-butoxycarbonylethyl, hydroxycarbonylmethyl, hydroxycarbonylethyl, hydroxycarbonyl, methylaminocarbonylmethyl, ethylaminocarbonylmethyl, n-propylaminocarbonylmethyl, isopropylaminocarbonylmethyl, benzylaminocarbonylmethyl, phenylaminocarbonylmethyl, cyclopropylaminocarbonylmethyl, cyclobutylaminocarbonylmethyl, cyclopentylaminocarbonylmethyl, cyclohexylaminocarbonylmethyl, dimethylaminocarbonylmethyl, diethylaminocarbonylmethyl, allylaminocarbonylmethyl, methylaminomethyl, dimethylaminomethyl, N-propylaminocarbonylmethyl, Diethylaminomethyl, ethylaminomethyl, isopropylaminomethyl, N-propylaminomethyl, N-butylaminomethyl, methylaminoethyl, dimethylaminoethyl, diethylaminoethyl, N-pyrrolidinylmethyl, N-piperidinylmethyl, hydroxyimino, methoxyimino, ethoxyimino, N-propoxylimino, N-butoxyimino, isopropoxyimino, tert-butoxyimino, cyclopropylmethoxyimino, cyclobutylmethoxyimino, cyclopentylmethoxyimino, cyclohexylmethoxyimino, benzyloxyimino, phenoxyimino, allyloxyimino, p-Cl-phenylmethoxyimino, phenylethynyl, p-Cl-phenylethynyl, m-Cl-phenylethynyl, o-Cl-phenylethynyl, p-Cl-phenylethynyl, N-propylaminoethyl, N-pyrrolidinylmethyl, N-piperidinylmethyl, N-hydroxyimino, methoxyimino, cyclohexylmethoxyimino, benzyloxy, p-F-phenylethynyl, m-F-phenylethynyl, o-F-phenylethynyl, pyridin-2-ylethynyl, pyridin-3-ylethynyl, thien-2-ylethynyl, trimethylsilylethynyl, triethylsilylethynyl, tris (isopropyl) silylethynyl, cyclopropylethynyl, cyclobutylethynyl, cyclopentylethynyl, cyclohexylethynyl, phenyl, benzyl, p-Cl-phenyl, m-Cl-phenyl, o-Cl-phenyl, p-F-phenyl, m-F-phenyl, o-F-phenyl, p-trifluoromethylphenyl, m-trifluoromethylphenyl, o-trifluoromethylphenyl, p-methylphenyl, m-methylphenyl, o-methylahenyl, o-methylanyl, p-methylanyl, P-methoxyphenyl, m-methoxyphenyl, o-methoxyphenyl, p-Cl-phenylmethyl, m-Cl-phenylmethyl, o-Cl-phenylmethyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, thiophen-2-yl, thiophen-3-yl, furan-2-yl, furan-3-yl, pyrimidin-2-yl, pyrazin-2-yl, methoxymethoxymethyl, ethoxymethyl, methoxyethoxymethyl, methylaminosulfonylamino, dimethylaminosulfonylamino, ethylaminosulfonylamino, diethylaminosulfonylamino, isopropylaminosulfonylamino, cyclopropylaminosulfonylamino, cyclobutylaminosulfonylamino, cyclopentylaminosulfonylamino, p-Cl-phenylmethyl, o-Cl-phenylmethyl, furan-2-yl, pyrimidin-2-yl, ethoxymethyl, methoxyethoxymethyl, methylaminosulfonylamino, dimethylaminosulfonylamino, ethylamino, Cyclohexylaminosulfonylamino, diazo, phenyldiazo, trimethylsilyl, tris (isopropyl) silyl, triethylsilyl, dimethyl (phenyl) silyl, diphenyl (methyl) silyl,
R14And R15Independently of one another, represents hydrogen, methyl, ethyl, n-propyl, isopropyl, n-butyl, fluorine, or
R9And R15Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
and
w represents oxygen.
5. A compound of the general formula (I) and/or a salt thereof as claimed in claim 1, characterized in that
R1Represents hydrogen, methyl, ethyl, n-propyl, 1-methylethyl, n-butyl, 1-methylprop-1-yl, 2-methylprop-1-yl, 1-dimethylethyl-1-yl, n-pentyl, 1-methylbut-1-yl, 2-methylbut-1-yl, 3-methylbut-1-yl, 1-dimethylprop-1-yl, 1, 2-dimethylprop-1-yl, 2-dimethylprop-1-yl, 1-ethylprop-1-yl, n-hexyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1-dimethylbutyl, 1, 2-dimethylbutyl, 1, 3-dimethylbutyl, 2, 2-dimethylbutyl, 2, 3-dimethylbutyl, 3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1, 2-trimethylpropyl, 1,2, 2-trimethylpropyl, 1-ethyl-1-methylpropyl, 1-ethyl-2-methylpropyl, trifluoromethyl, pentafluoroethyl, 1,2, 2-tetrafluoroethyl, heptafluoro-n-propyl, heptafluoroisopropyl, nonafluorobutyl, chlorodifluoromethyl, bromodifluoromethyl, dichlorofluoromethyl, iododifluoromethyl, bromofluoromethyl, 1-fluoroethyl, 2-fluoroethyl, fluoromethyl, difluoromethyl, 2, 2-difluoroethyl, 2,2, 2-trifluoroethyl, 2, 3-dimethylbutyl, 1,2, 2-trimethylpropyl, 1-ethyl-1-methylpropyl, 1-ethyl-2-methylpropyl, trifluoromethyl, iododifluoromethyl, bromofluoromethyl, 2-fluoroethyl, 2-, 3,3, 3-trifluoropropan-1-yl, 3,3, 3-trifluoropropan-2-yl, difluoro-tert-butyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, adamantan-1-yl, adamantan-2-yl, 1-methylcyclopropyl, 2-dimethylcyclopropyl, 2, 3-dimethylcyclopropyl, 1 '-bis (cyclopropyl) -1-yl, 1' -bis (cyclopropyl) -2-yl, 2 '-methyl-1, 1' -bis (cyclopropyl) -2-yl, 1-cyanocyclopropyl, 2-cyanopropylamino, 2-fluoropropylamino, 1-methylcyclobutyl, 2-methylcyclobutyl, 3-methylcyclobutyl, 1-cyanocyclobutyl, 2-cyanocyclobutyl, 3-cyanocyclobutyl, 1-allylcyclopropyl, 1-vinylcyclobutyl, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 1-methoxycyclohexyl, 2-methoxycyclohexyl, 3-methoxycyclohexyl, cyclopropylmethyl, cyclobutylmethyl, cyclopentylmethyl, cyclohexylmethyl, phenyl, p-F-phenyl, m-F-phenyl, o-F-phenyl, p-Cl-phenyl, m-Cl-phenyl, o-Cl-phenyl, p-Cl-cyclohexyl, p-cyclohexyl, 1-vinylcyclopropyl, 1-vinylcyclobutyl, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, cyclopropylmethyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, thiophen-2-yl, thiophen-3-yl, furan-2-yl, furan-3-yl, tetrahydrofuran-2-yl, tetrahydrofuran-3-yl, benzyl, p-Cl-benzyl, p-F-benzyl, p-methoxybenzyl, p-methylbenzyl, p-trifluoromethylbenzyl, p-nitrobenzyl, m-Cl-benzyl, m-F-benzyl, m-methoxybenzyl, m-methylbenzyl, o-Cl-benzyl, o-F-benzyl, o-methoxybenzyl, o-methylbenzyl, 1-phenyleth-1-yl, o-methoxybenzyl, o-methylbenzyl, o-phenyleth-1-yl, o-methyl-benzyl, p-nitrobenzyl, m-benzyl, m-F-benzyl, 2-Phenylethan-1-yl, 1- (o-chlorophenyl) ethan-1-yl, 1- (o-fluorophenyl) ethan-1-yl, 1- (o-methylphenyl) ethan-1-yl, 1- (o-bromophenyl) ethan-1-yl, 1- (o-iodophenyl) ethan-1-yl, pyridin-2-ylmethyl, pyridin-3-ylmethyl, pyridin-4-ylmethyl, pyrimidin-2-ylmethyl, pyrimidin-4-ylmethyl, tetrahydrofuran-2-ylmethyl, o-cyanophenylmethyl, m-cyanophenylmethyl, p-cyanophenylmethyl, cyanomethyl, cyanoethyl, methoxycarbonyl, ethoxycarbonyl, n-propoxycarbonyl, isopropoxycarbonyl, iso-propoxycarbonyl, Tert-butoxycarbonyl, benzyloxycarbonyl, allyloxycarbonyl, methylcarbonyl, ethylcarbonyl, n-propylcarbonyl, isopropylcarbonyl, n-butylcarbonyl, 1-methylprop-1-ylcarbonyl, 2-methylprop-1-ylcarbonyl, 1-dimethyleth-1-ylcarbonyl, phenylcarbonyl, methylaminocarbonyl, dimethylaminocarbonyl, ethylaminocarbonyl, n-propylaminocarbonyl, isopropylaminocarbonyl, n-butylaminocarbonyl, tert-butylaminocarbonyl, benzylaminocarbonyl, methoxycarbonylmethyl, ethoxycarbonylmethyl, tert-butoxycarbonylmethyl, benzyloxycarbonylmethyl, methoxycarbonylethyl, ethoxycarbonylethyl, tert-butoxycarbonylmethyl, benzyloxycarbonylmethyl, ethoxycarbonylethyl, tert-butoxycarbonylmethyl, benzyloxycarbonyl Alkylcarbonylmethyl, methylcarbonyloxymethyl, ethylcarbonyloxymethyl, n-propylcarbonyloxymethyl, 1-methylethylcarbonyloxymethyl, 1-dimethylethylcarbonyloxymethyl, hydroxycarbonylmethyl, hydroxycarbonylethyl, hydroxycarbonyln-propyl, methoxy, ethoxy, n-propoxy, isopropoxy, methoxymethyl, ethoxymethyl, n-propoxymethyl, isopropoxymethyl, n-butoxymethyl, methoxyethyl, ethoxyethyl, n-propoxyethyl, isopropoxyethyl, methoxy-n-propyl, ethoxy-n-propyl, methoxy-n-butyl, amino, dimethylamino, methyl (ethyl) amino, diethylamino, cyanomethyl, cyanoethyl, prop-2-yn-1-yl,
R2and R9Independently of one another, represents hydrogen, hydroxy, fluorine, methyl, ethyl, n-propyl, isopropyl, n-butyl, 1-methylprop-1-yl, 2-methylprop-1-yl, 1-dimethyleth-1-yl, trifluoromethyl, difluoromethyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, phenyl, p-F-phenyl, m-F-phenyl, o-F-phenyl, p-Cl-phenyl, m-Cl-phenyl, o-Cl-phenyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, thiophen-2-yl, thiophen-3-yl, furan-2-yl, methyl, ethyl, propyl, isopropyl, n-butyl, 1-methylprop-1-yl, 2-methylprop-1-yl, 1-dimethyleth-1-yl, trifluoromethyl, difluoromethyl, cyclopropyl, cyclobutyl, Furan-3-yl, methoxymethyl, ethoxymethyl, methoxyethyl, ethoxyethyl, methoxy, ethoxy, n-propoxy, isopropoxy, trifluoromethoxy, difluoromethoxy, methylthio, ethylthio, trifluoromethylthio, dimethylamino, methylamino, diethylamino, methyl (ethyl) amino, cyano, or
R1And R2Together with the nitrogen or carbon atom to which they are respectively attached form a fully or partially saturated ring having a total of 3 to 7 members, said ring being optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted, or
R2And R9Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted，
R3Represents hydroxy, mercapto, fluoro, chloro, bromo, iodo, methoxy, ethoxy, n-propoxy, 1-methylethoxy, n-butoxy, 1-methylpropoxy, 2-methylpropoxy, 1-dimethylethoxy, n-pentyloxy, 1-methylbutoxy, 2-methylbutoxy, 3-methylbutoxy, 1-dimethylpropoxy, 1, 2-dimethylpropoxy, 2-dimethylpropoxy, 1-ethylpropoxy, n-hexyloxy, 1-methylpentyloxy, 2-methylpentyloxy, 3-methylpentyloxy, 4-methylpentyloxy, 1-dimethylbutyloxy, 1, 2-dimethylbutyloxy, 1, 3-dimethylbutyloxy, 2-dimethylbutyloxy, n-butyloxy, 1-methylpropyloxy, 2-methylbutoxy, 3-methylbutoxy, 2, 3-dimethylbutoxy, 3-dimethylbutoxy, 1-ethylbutoxy, 2-ethylbutoxy, 1, 2-trimethylpropoxy, 1,2, 2-trimethylpropoxy, 1-ethyl-1-methylpropoxy, 1-ethyl-2-methylpropoxy, cyclopropylmethoxy, cyclobutylmethoxy, cyclopentylmethoxy, cyclohexylmethoxy, benzyloxy, p-chlorophenylmethoxy, m-chlorophenylmethoxy, o-chlorophenylmethoxy, p-methoxyphenylmethoxy, p-nitrophenylmethoxy, methoxymethoxy, methoxyethoxy, methoxy-n-propoxy, methoxy-n-butoxy, ethoxymethoxy, ethoxyethoxy, ethoxy-n-propoxy, ethoxy-n-butoxy, n-propoxy, methoxy-n-propoxy, n-butoxy, n-propoxy-methoxy-propoxy, n-butoxy, Isopropoxymethoxy group, methylcarbonyloxy group, ethylcarbonyloxy group, n-propylcarbonyloxy group, 1-methylethylcarbonyloxy group, n-butylcarbonyloxy group, 1-methylpropylcarbonyloxy group, 2-methylpropylcarbonyloxy group, 1-dimethylethylcarbonyloxy group, n-pentylcarbonyloxy group, 1-methylbutylcarbonyloxy group, 2-methylbutylcarbonyloxy group, 3-methylbutylcarbonyloxy group, 1-dimethylpropylcarbonyloxy group, 1, 2-dimethylpropylcarbonyloxy group, 2-dimethylpropylcarbonyloxy group, 1-ethylpropylcarbonyloxy group, n-hexylcarbonyloxy group, 1-methylpentylcarbonyloxy group, 2-methylpentylcarbonyloxy group, 3-methylpentylcarbonyloxy group, 4-methylpentylcarbonyloxy group, n-propylcarbonyloxy group, n-butylcarbonyloxy group, 1-methylbutylcarbonyloxy group, 1-methylpropylc, 1, 1-dimethylbutylcarbonyloxy, 1, 2-dimethylbutylcarbonyloxy, 1, 3-dimethylbutylcarbonyloxy, 2-dimethylbutylcarbonyloxy, 2, 3-dimethylbutylcarbonyloxy, 3-dimethylbutylcarbonyl Oxy, 1-ethylbutylcarbonyloxy, 2-ethylbutylcarbonyloxy, 1, 2-trimethylpropylcarbonyloxy, 1,2, 2-trimethylpropylcarbonyloxy, 1-ethyl-1-methylpropylcarbonyloxy, 1-ethyl-2-methylpropylcarbonyloxy, phenylcarbonyloxy, p-chlorophenylcarbonyloxy, m-chlorophenylcarbonyloxy, o-chlorophenylcarbonyloxy, p-fluorophenylcarbonyloxy, m-fluorophenylcarbonyloxy, o-fluorophenylcarbonyloxy, benzylcarbonyloxy, thien-2-ylcarbonyloxy, furan-2-ylcarbonyloxy, cyclopropylcarbonyloxy, cyclobutylcarbonyloxy, cyclopentylcarbonyloxy, cyclohexylcarbonyloxy, 1-fluorocycloprop-1-ylcarbonyloxy, o, 1-chlorocycloprop-1-ylcarbonyloxy, 1-cyanocycloprop-1-ylcarbonyloxy, 1-methylcycloprop-1-ylcarbonyloxy, 1-trifluoromethylcycloprop-1-ylcarbonyloxy, adamantylcarbonyloxy, trifluoromethylcarbonyloxy, difluoromethylcarbonyloxy, methoxycarbonyloxy, ethoxycarbonyloxy, n-propoxycarbonyloxy, isopropoxycarbonyloxy, n-butoxycarbonyloxy, 1-dimethylethoxycarbonyl-oxy, 2-dimethylpropoxycarbonyloxy, benzyloxycarbonyloxy, allyloxycarbonyloxy, cyclopropyloxycarbonyloxy, cyclobutyloxycarbonyloxy, cyclopentyloxycarbonyloxy, cyclohexyloxycarbonyloxy, cyclopropylmethoxycarbonyloxy, cyclobutylmethoxycarbonyloxy, cyclobutyloxycarbonyloxy, and the like, Cyclopentylmethoxycarbonyloxy, cyclohexylmethoxycarbonyloxy, 3,3, 3-trifluoroethoxycarbonyloxy, 2-difluoroethoxycarbonyloxy, pyridin-2-ylcarbonyloxy, pyridin-3-ylcarbonyloxy, pyridin-4-ylcarbonyloxy, 4-trifluoromethylpyridin-3-ylcarbonyloxy, allylcarbonyloxy, methylsulfonyloxy, ethylsulfonyloxy, n-propylsulfonyloxy, 1-methylethylsulfonyloxy, cyclopropylsulfonyloxy, cyclobutylsulfonyloxy, cyclopentylsulfonyloxy, cyclohexylsulfonyloxy, phenylsulfonyloxy, p-chlorophenylsulfonyloxy, m-chlorophenylsulfonyloxy, o-chlorophenylsulfonyloxy, p-fluorophenylsulfonyloxy, m-fluorophenylsulfonyloxy, o-fluorophenylsulfonyloxy, 2-difluoroethoxycarbonyloxy, pyridine-2-ethylsulfonyloxy, n-propylsulfonyloxy, n-, P-methoxyphenyl sulfonyloxy, m-methoxyphenyl sulfonyloxy, o-methoxyphenyl sulfonyloxy, p-methylphenyl sulfonyloxy, m-methylphenyl Arylsulfonyloxy, o-methylphenylsulfonyloxy,
R6represents hydrogen, and is selected from the group consisting of,
R14and R15Independently of one another, represents hydrogen, methyl, ethyl, n-propyl, isopropyl, n-butyl, fluorine, or
R9And R15Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
w represents oxygen, and W represents oxygen,
and
q represents one of the moieties Q-1.1 to Q-30.5 specified hereinafter, wherein the arrow represents the bond of the respective Q group to the nitrogen of the tetrahydropyrimidinone of the general formula (I)
6. A compound of the general formula (I) and/or a salt thereof as claimed in claim 1, characterized in that
R1Represents hydrogen, methyl, ethyl, n-propyl, 1-methylethyl, n-butyl, 1-methylprop-1-yl, 2-methylprop-1-yl, 1-dimethylethyl-1-yl, n-pentyl, 1-methylbut-1-yl, 2-methylbut-1-yl, 3-methylbut-1-yl, 1-dimethylprop-1-yl, 1, 2-dimethylprop-1-yl, 2-dimethylprop-1-yl, 1-ethylprop-1-yl, n-hexyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1-dimethylbutyl, 1, 2-dimethylbutyl, 1, 3-dimethylbutyl, 2, 2-dimethylbutyl, 2, 3-dimethylbutyl, 3-dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1, 2-trimethylpropyl, 1,2, 2-trimethylpropyl, 1-ethyl-1-methylpropyl, 1-ethyl-2-methylpropyl Trifluoromethyl, difluoromethyl, 2, 2-difluoroethyl, 2,2, 2-trifluoroethyl, 3,3, 3-trifluoroprop-1-yl, 3,3, 3-trifluoroprop-2-yl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, adamantan-1-yl, adamantan-2-yl, 1-methylcyclopropyl, 2, 2-dimethylcyclopropyl, 2, 3-dimethylcyclopropyl, 1-cyanocyclopropyl, 2-cyanocyclopropyl, 1-methylcyclobutyl, 2-methylcyclobutyl, 3-methylcyclobutyl, 1-cyanocyclobutyl, 2-cyanocyclobutyl, 3-cyanocyclobutyl, 1-allylcyclopropyl, 1-vinylcyclobutyl, 2-fluoropropyl, 3-fluoropropyl, 2-fluorop, 1-vinylcyclopropyl, 1-ethylcyclopropyl, 1-methylcyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 1-methoxycyclohexyl, 2-methoxycyclohexyl, 3-methoxycyclohexyl, cyclopropylmethyl, cyclobutylmethyl, cyclopentylmethyl, cyclohexylmethyl, phenyl, p-F-phenyl, m-F-phenyl, o-F-phenyl, p-Cl-phenyl, m-Cl-phenyl, o-Cl-phenyl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, thiophen-2-yl, thiophen-3-yl, furan-2-yl, methyl ethyl, propyl, butyl, furan-3-yl, tetrahydrofuran-2-yl, tetrahydrofuran-3-yl, benzyl, p-Cl-benzyl, p-F-benzyl, p-methoxybenzyl, p-methylbenzyl, p-trifluoromethylbenzyl, p-nitrobenzyl, m-Cl-benzyl, m-F-benzyl, m-methoxybenzyl, m-methylbenzyl, o-Cl-benzyl, o-F-benzyl, o-methoxybenzyl, o-methylbenzyl, 1-phenyleth-1-yl, 2-phenyleth-1-yl, 1- (o-chlorophenyl) eth-1-yl, 1- (o-fluorophenyl) eth-1-yl, 1- (o-methylphenyl) eth-1-yl, 1- (o-bromophenyl) eth-1-yl, benzyl, p-methylbenzyl, p-trifluoromethylbenzyl, p-nitrobenzyl, m-Cl-benzyl, m-F-, 1- (o-iodophenyl) eth-1-yl, pyridin-2-ylmethyl, pyridin-3-ylmethyl, pyridin-4-ylmethyl, pyrimidin-2-ylmethyl, pyrimidin-4-ylmethyl, tetrahydrofuran-2-ylmethyl, o-cyanophenylmethyl, m-cyanophenylmethyl, p-cyanophenylmethyl, cyanomethyl, cyanoethyl, methoxycarbonyl, ethoxycarbonyl, n-propoxycarbonyl, isopropoxycarbonyl, t-butoxycarbonyl, benzyloxycarbonyl, allyloxycarbonyl, methylcarbonyl, ethylcarbonyl, n-propylcarbonyl, isopropylcarbonyl, n-butylcarbonyl, 1-methylpropan-1-ylcarbonyl, 2-methylpropan-1-ylcarbonyl, 1-dimethylethyl-1-ylcarbonyl, pyridine-4-ylmethyl, pyrimidin-2-ylmethyl, pyridine-2-ylmethyl, pyridylcarbonyl, isopropylcarbonyl, benzyloxycarbonyl, allyloxycarbonyl, methylcarbonyl, ethylcarbonyl, n-propylcarbonyl, isopropylcarbonyl, Phenylcarbonyl, methylaminocarbonyl, dimethyl Alkylaminocarbonyl, ethylaminocarbonyl, n-propylaminocarbonyl, isopropylaminocarbonyl, n-butylaminocarbonyl, tert-butylaminocarbonyl, benzylaminocarbonyl, methoxycarbonylmethyl, ethoxycarbonylmethyl, tert-butoxycarbonylmethyl, benzyloxycarbonylmethyl, methoxycarbonylethyl, ethoxycarbonylethyl, tert-butoxycarbonylmethyl, benzyloxycarbonylmethyl, methylcarbonyloxymethyl, ethylcarbonyloxymethyl, n-propylcarbonyloxymethyl, 1-methylethylcarbonyloxymethyl, 1-dimethylethylcarbonyloxymethyl, hydroxycarbonylmethyl, hydroxycarbonylethyl, hydroxycarbonyl-n-propyl, methoxy, ethoxy, n-propoxy, isopropoxy, methoxymethyl, ethoxymethyl, n-propoxymethyl, isopropoxymethyl, n-butoxymethyl, methoxyethyl, ethoxymethyl, n-propoxymethyl, n-butoxymethyl, ethoxycarbonylmethyl, n-butyloxycarbonyl, tert-butyl, Ethoxyethyl, n-propoxyethyl, isopropoxyethyl, methoxy-n-propyl, ethoxy-n-propyl, methoxy-n-butyl, amino, dimethylamino, methyl (ethyl) amino, diethylamino, cyanomethyl, prop-2-yn-1-yl,
R2and R9Independently of one another, represents hydrogen, fluorine, methyl, ethyl, n-propyl, isopropyl, n-butyl, 1-methylprop-1-yl, 2-methylprop-1-yl, 1-dimethyleth-1-yl, trifluoromethyl, difluoromethyl, cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl, methoxymethyl, ethoxymethyl, methoxyethyl, ethoxyethyl, methoxy, ethoxy, n-propoxy, isopropoxy, trifluoromethoxy, difluoromethoxy, methylthio, ethylthio, trifluoromethylthio, dimethylamino, methylamino, diethylamino, methyl (ethyl) amino, or
R1And R2Together with the nitrogen or carbon atom to which they are respectively attached form a fully or partially saturated ring having a total of 3 to 7 members, said ring being optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted, or
R2And R9Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally substituted with 1 to 3A heteroatom spacer from N, O and S, and optionally further substituted,
R3represents hydroxy, mercapto, fluoro, chloro, bromo, iodo, methoxy, ethoxy, n-propoxy, 1-methylethoxy, n-butoxy, 1-methylpropoxy, 2-methylpropoxy, 1-dimethylethoxy, n-pentyloxy, 1-methylbutoxy, 2-methylbutoxy, 3-methylbutoxy, 1-dimethylpropoxy, 1, 2-dimethylpropoxy, 2-dimethylpropoxy, 1-ethylpropoxy, n-hexyloxy, 1-methylpentyloxy, 2-methylpentyloxy, 3-methylpentyloxy, 4-methylpentyloxy, 1-dimethylbutyloxy, 1, 2-dimethylbutyloxy, 1, 3-dimethylbutyloxy, 2-dimethylbutyloxy, n-butyloxy, 1-methylpropyloxy, 2-methylbutoxy, 3-methylbutoxy, 2, 3-dimethylbutoxy, 3-dimethylbutoxy, 1-ethylbutoxy, 2-ethylbutoxy, 1, 2-trimethylpropoxy, 1,2, 2-trimethylpropoxy, 1-ethyl-1-methylpropoxy, 1-ethyl-2-methylpropoxy, cyclopropylmethoxy, cyclobutylmethoxy, cyclopentylmethoxy, cyclohexylmethoxy, benzyloxy, p-chlorophenylmethoxy, m-chlorophenylmethoxy, o-chlorophenylmethoxy, p-methoxyphenylmethoxy, p-nitrophenylmethoxy, methoxymethoxy, methoxyethoxy, methoxy-n-propoxy, methoxy-n-butoxy, ethoxymethoxy, ethoxyethoxy, ethoxy-n-propoxy, ethoxy-n-butoxy, n-propoxy, methoxy-n-propoxy, n-butoxy, n-propoxy-methoxy-propoxy, n-butoxy, Isopropoxymethoxy group, methylcarbonyloxy group, ethylcarbonyloxy group, n-propylcarbonyloxy group, 1-methylethylcarbonyloxy group, n-butylcarbonyloxy group, 1-methylpropan-1-ylcarbonyloxy group, 2-methylpropan-1-ylcarbonyloxy group, 1-dimethyleth-1-ylcarbonyloxy group, n-pentylcarbonyloxy group, 1-methylbutylcarbonyloxy group, 2-methylbutylcarbonyloxy group, 3-methylbutylcarbonyloxy group, 1-dimethylpropylcarbonyloxy group, 1, 2-dimethylpropylcarbonyloxy group, 2-dimethylpropylcarbonyloxy group, 1-ethylpropylcarbonyloxy group, n-hexylcarbonyloxy group, 1-methylpentylcarbonyloxy group, 2-methylpentylcarbonyloxy group, 3-methylpentylcarbonyloxy group, 2-methylpentylcarbonyloxy group, n-, 4-methylpentylcarbonyloxy, 1-dimethylbutylcarbonyloxy, 1, 2-dimethylbutylcarbonyloxy, 1, 3-dimethylbutylcarbonyloxy, 2-dimethylbutyl Carbonyloxy, 2, 3-dimethylbutylcarbonyloxy, 3-dimethylbutylcarbonyloxy, 1-ethylbutylcarbonyloxy, 2-ethylbutylcarbonyloxy, 1, 2-trimethylpropylcarbonyloxy, 1,2, 2-trimethylpropylcarbonyloxy, 1-ethyl-1-methylpropylcarbonyloxy, 1-ethyl-2-methylpropylcarbonyloxy, phenylcarbonyloxy, p-chlorophenylcarbonyloxy, m-chlorophenylcarbonyloxy, o-chlorophenylcarbonyloxy, p-fluorophenylcarbonyloxy, m-fluorophenylcarbonyloxy, o-fluorophenylcarbonyloxy, benzylcarbonyloxy, thien-2-ylcarbonyloxy, furan-2-ylcarbonyloxy, cyclopropylcarbonyloxy, cyclobutylcarbonyloxy, tert-butylcarbonyloxy, 2-ethylbutylcarbonyloxy, 1-ethyl-2-methylpropylcarbonyloxy, 1-, Cyclopentylcarbonyloxy, cyclohexylcarbonyloxy, 1-fluorocycloprop-1-ylcarbonyloxy, 1-chlorocycloprop-1-ylcarbonyloxy, 1-cyanocycloprop-1-ylcarbonyloxy, 1-methylcycloprop-1-ylcarbonyloxy, 1-trifluoromethylcycloprop-1-ylcarbonyloxy, adamantylcarbonyloxy, trifluoromethylcarbonyloxy, difluoromethylcarbonyloxy, methoxycarbonyloxy, ethoxycarbonyloxy, n-propoxycarbonyloxy, isopropoxycarbonyloxy, n-butoxycarbonyloxy, 1-dimethylethoxycarbonyl-oxy, 2-dimethylpropoxycarbonyloxy, benzyloxycarbonyloxy, allyloxycarbonyloxy, cyclopropyloxycarbonyloxy, cyclobutyloxycarbonyloxy, and the like, Cyclopentyloxycarbonyloxy, cyclohexyloxycarbonyloxy, cyclopropylmethoxycarbonyloxy, cyclobutylmethoxycarbonyloxy, cyclopentylmethoxycarbonyloxy, cyclohexylmethoxycarbonyloxy, 3,3, 3-trifluoroethoxycarbonyloxy, 2-difluoroethoxycarbonyloxy, pyridin-2-ylcarbonyloxy, pyridin-3-ylcarbonyloxy, pyridin-4-ylcarbonyloxy, 4-trifluoromethylpyridin-3-ylcarbonyloxy, allylcarbonyloxy, methylsulfonyloxy, ethylsulfonyloxy, n-propylsulfonyloxy, 1-methylethylsulfonyloxy, cyclopropylsulfonyloxy, cyclobutylsulfonyloxy, cyclopentylsulfonyloxy, cyclohexylsulfonyloxy, phenylsulfonyloxy, p-chlorophenylsulfonyloxy, m-chlorophenylsulfonyloxy, cyclobutylsulfonyloxy, cyclopentylsulfonyloxy, cyclohexylsulfonyloxy, p-chlorophenylsulfonyloxy, m-chlorophenylsulfonyloxy, cyclopentylsulfonyloxy, cyclopentylsulf, O-chlorophenylsulfonyloxy, p-fluorophenylsulfonyloxy, m-fluorophenylsulfonyloxy, o-fluorophenylsulfonyloxy, p-methoxyphenylsulfonyloxy, m-methoxyphenylsulfonyloxy, O-methoxyphenylsulfonyloxy, p-methylphenylsulfonyloxy, m-methylphenylsulfonyloxy, o-methylphenylsulfonyloxy,
R6represents hydrogen, and is selected from the group consisting of,
R14and R15Independently of one another, represents hydrogen, methyl, ethyl, n-propyl, isopropyl, n-butyl, fluorine, or
R9And R15Together with the carbon atom to which they are each attached form a fully or partially saturated ring having a total of 3 to 7 members, optionally interrupted by 1 to 3 heteroatoms selected from N, O and S, and optionally further substituted,
w represents oxygen, and W represents oxygen,
and
q represents one of the moieties Q-1.1 to Q-30.5 as described in claim 5.
7. Use of one or more compounds of the general formula (I) and/or salts thereof as defined in any of claims 1 to 6 as herbicides and/or plant growth regulators, preferably in crops of useful plants and/or ornamental plants.
8. A herbicidal and/or plant growth regulating composition, characterized in that the composition comprises one or more compounds of formula (I) and/or salts thereof, as defined in any one of claims 1 to 6, and one or more further substances selected from the group (I) and/or (ii), wherein
(i) One or more further agrochemical active substances, preferably selected from insecticides, acaricides, nematicides, further herbicides, fungicides, safeners, fertilizers and/or further growth regulators,
(ii) One or more formulation auxiliaries customary in crop protection.
9. A method for controlling harmful plants or for regulating the growth of plants, characterized in that an effective amount of
-one or more compounds of formula (I) and/or salts thereof, as defined in any one of claims 1 to 6, or
-a composition as claimed in claim 8,
to the plant, to the seed of the plant, to the soil or to the area of cultivation in or on which the plant is growing.
Example Nos. I.1 to 72
1H-NMR(400MHz,CDCl3,ppm)6.51(s,1H),5.69(m,1H),3.83(m,1H),3.21(m,1H9,3.06(s,3H),2.33(s,3H),2.19-2.16(m,2H)。